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Thalidomide-NH-PEG1-NH-Boc

Product Name
Thalidomide-NH-PEG1-NH-Boc
CAS No.
2154342-17-1
Chemical Name
Thalidomide-NH-PEG1-NH-Boc
Synonyms
Thalidomide-NH-PEG1-NH-Boc;Thalidomide-4-NH-PEG1-NH-Boc;Thalidomide-4-NH-PEG1-C2-NH-Boc;tert-butyl (2-(2-((2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)amino)ethoxy)ethyl)carbamate;Carbamic acid, N-[2-[2-[[2-(2,6-dioxo-3-piperidinyl)-2,3-dihydro-1,3-dioxo-1H-isoindol-4-yl]amino]ethoxy]ethyl]-, 1,1-dimethylethyl ester
CBNumber
CB011336433
Molecular Formula
C22H28N4O7
Formula Weight
460.48
MOL File
2154342-17-1.mol
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Thalidomide-NH-PEG1-NH-Boc Property

Boiling point:
715.3±60.0 °C(Predicted)
Density 
1.346±0.06 g/cm3(Predicted)
pka
10.74±0.40(Predicted)
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Hazard and Precautionary Statements (GHS)

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Thalidomide-NH-PEG1-NH-Boc Chemical Properties,Usage,Production

Uses

Thalidomide-4-NH-PEG1-NH-Boc is a Boc-modified Thalidomide (HY-14658) that acts as a Cereblon ligand to recruit CRBN protein. The Boc protecting group at the end of Thalidomide-4-NH-PEG1-NH-Boc can be removed under acidic conditions to participate in the synthesis of PROTAC molecules. Thalidomide-4-NH-PEG1-NH-Boc is a key intermediate in the synthesis of CRBN-based PROTAC molecules.

IC 50

Cereblon

References

[1] Fischer ES, et al. Structure of the DDB1-CRBN E3 ubiquitin ligase in complex with thalidomide. Nature. 2014 Aug 7;512(7512):49-53.??[Content Brief] DOI:10.1038/nature13527

Thalidomide-NH-PEG1-NH-Boc Preparation Products And Raw materials

Raw materials

Preparation Products

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Thalidomide-NH-PEG1-NH-Boc Suppliers

Daicel Chiral Technologies (China)CO.,LTD
Tel
021-50460086-9 15921403865
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+86-21-50462321
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han_yajun@dctc.daicel.com
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China
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7471
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65
CR Corporation Limited
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+8613062833949
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fred.wen@crcorporation.cn
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China
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8645
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Zhengzhou Convergence Chemical Co. LTD
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0371-0371-53736046 13393710386
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QQ:2853979814
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2853979814@qq.com
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China
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9947
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Shandong Territorial sea Biological Technology Co., LTD
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15092083467
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18660263263@163.com
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China
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2810
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Xi'an Qiyue Biotechnology Co., Ltd.
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400-400-6966-012-012 17778955912
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2957605606@qq.com
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China
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2535
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Chengdu Yuxin Technology Co., Ltd.
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13558691827
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yuxinpharma@126.com
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China
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Shanghai Hongboshangyi Pharmaceutical Technology Co. , Ltd.
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15927323052
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shenqianyan@prssh.com
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China
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999
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Suzhou Haiben Pharmaceutical Co., Ltd
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19353112242
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1816280386@qq.com
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China
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8045
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Shanghai Yifei Biotechnology Co. , Ltd.
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021-65675885 18964387627
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customer_service@efebio.com
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China
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11973
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58
Jilin Chinese Academy of Sciences-yanshen Technology
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18143011203
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ET-market@chemextension.com
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China
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32034
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58
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View Lastest Price from Thalidomide-NH-PEG1-NH-Boc manufacturers

Shaanxi Dideu New Materials Co. Ltd
Product
Thalidomide-NH-PEG1-NH-Boc 2154342-17-1
Price
US $0.00/kg
Min. Order
1kg
Purity
99%
Supply Ability
10000KGS
Release date
2025-03-08