Ceefourin 1
- Product Name
- Ceefourin 1
- CAS No.
- 315702-40-0
- Chemical Name
- Ceefourin 1
- Synonyms
- Ceefourin 1;Ceefourin 1, 10 mM in DMSO;Ceefourin 1, MRP4 inhibitor;5-[(2-Benzothiazolylthio)methyl]-2,4-dihydro-4-methyl-3H-1,2,4-triazole-3-thione;3H-1,2,4-Triazole-3-thione, 5-[(2-benzothiazolylthio)methyl]-2,4-dihydro-4-methyl-;P-glycoprotein,chemosensitizers,inhibit,efflux,protein,resistance,Ceefourin 1,Ceefourin1,MRP4,HEK293,D-luciferin,ABC,ABCG2,P-gp,multidrug,MRP1,Inhibitor,neuroblastoma,Ceefourin-1,ABCC1,BCRP
- CBNumber
- CB33152938
- Molecular Formula
- C11H10N4S3
- Formula Weight
- 294.42
- MOL File
- 315702-40-0.mol
Ceefourin 1 Property
- Melting point:
- 181° - 182°C
- Boiling point:
- 422.1±55.0 °C(Predicted)
- Density
- 1.58±0.1 g/cm3(Predicted)
- storage temp.
- -20°C, Inert atmosphere
- solubility
- Chloroform (Slightly), Methanol (Slightly, Heated)
- form
- Solid
- pka
- 8.37±0.20(Predicted)
- color
- Pale Yellow
Hazard and Precautionary Statements (GHS)
- Symbol(GHS)
-
- Signal word
- Warning
- Hazard statements
-
H315Causes skin irritation
H319Causes serious eye irritation
- Precautionary statements
-
P264Wash hands thoroughly after handling.
P264Wash skin thouroughly after handling.
P280Wear protective gloves/protective clothing/eye protection/face protection.
P302+P352IF ON SKIN: wash with plenty of soap and water.
P305+P351+P338IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses, if present and easy to do. Continuerinsing.
P332+P313IF SKIN irritation occurs: Get medical advice/attention.
P337+P313IF eye irritation persists: Get medical advice/attention.
N-Bromosuccinimide Price
- Product number
- SML3334
- Product name
- Ceefourin 1
- Purity
- ≥95% (HPLC)
- Packaging
- 5MG
- Price
- $63.27
- Updated
- 2025/07/31
- Product number
- SML3334
- Product name
- Ceefourin 1
- Purity
- ≥95% (HPLC)
- Packaging
- 25MG
- Price
- $268
- Updated
- 2025/07/31
- Product number
- 5867
- Product name
- Ceefourin1
- Purity
- ≥98%(HPLC)
- Packaging
- 10
- Price
- $169
- Updated
- 2021/12/16
- Product number
- 5867
- Product name
- Ceefourin1
- Purity
- ≥98%(HPLC)
- Packaging
- 50
- Price
- $711
- Updated
- 2021/12/16
- Product number
- C231350
- Product name
- Ceefourin1
- Packaging
- 50mg
- Price
- $565
- Updated
- 2021/12/16
Ceefourin 1 Chemical Properties,Usage,Production
Uses
Ceefourin 1 inhibit the transport of a broad range of multidrug resistance-associated protein 4 (MRP4).
Biological Activity
Ceefourin 1 is a potent and highly selective MRP4 (Multidrug resistance protein 4) inhibitor th at exhibits low cellular toxicity and high microsomal and acid stability. Ceefourin 1 inhibits PDAC (pancreatic ductal adenocarcinoma) cell proliferation through MRP4-dependent cAMP extrusion thereby activation of the cAMP/Epac/Rap1 signaling pathway.
storage
Store at +4°C