GSK 2801

ChemicalBook > CAS DataBase List > GSK 2801

Product Name: GSK 2801
CAS No.: 1619994-68-1
Chemical Name: GSK 2801
Synonyms: CS-1607;GSK2801;GSK 280;GSK 2801;GSK-2801;GSK2801, >98%;GSK-2801; GSK 280;GSK2801 GSK-2801;GSK2801;GSK-2801;GSK 2801;1-[1-[2-(Methylsulfonyl)phenyl]-7-propoxy-3-indolizinyl]ethanone
CBNumber: CB52668513
Molecular Formula: C20H21NO4S
Formula Weight: 371.45
MOL File: 1619994-68-1.mol

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GSK 2801 Property

Density: 1.23±0.1 g/cm3(Predicted)
storage temp.: -20°C
solubility: insoluble in H2O; ≥18.55 mg/mL in DMSO; ≥2.82 mg/mL in EtOH with gentle warming and ultrasonic
form: solid
color: Light yellow to khaki

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Safety

Hazard Codes: Xn
Risk Statements: 22

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Hazard and Precautionary Statements (GHS)

Symbol(GHS)

Signal word

Warning

Hazard statements

H302Harmful if swallowed

Precautionary statements

P280Wear protective gloves/protective clothing/eye protection/face protection.

P305+P351+P338IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses, if present and easy to do. Continuerinsing.

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N-Bromosuccinimide Price

Cayman Chemical

Product number: 14120
Product name: GSK2801
Purity: ≥98%
Packaging: 1mg
Price: $32
Updated: 2024/03/01

Cayman Chemical

Product number: 14120
Product name: GSK2801
Purity: ≥98%
Packaging: 5mg
Price: $109
Updated: 2024/03/01

Tocris

Product number: 5635
Product name: GSK2801
Purity: ≥98%(HPLC)
Packaging: 10
Price: $160
Updated: 2021/12/16

TRC

Product number: G797680
Product name: GSK2801
Packaging: 25mg
Price: $335
Updated: 2021/12/16

TRC

Product number: G797680
Product name: GSK2801
Packaging: 1mg
Price: $55
Updated: 2021/12/16

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GSK 2801 Chemical Properties,Usage,Production

Description

BAZ2A/B are bromodomain-containing proteins whose biological function is believed to function similarly to ACF1, the Drosophila BAZ2B ortholog. ACF complexes play roles in establishing regular nucleosome spacing during chromatin assembly and influencing different remodeling outcomes at target loci. BAZ2A and BAZ2B constitute the central scaffolding protein of the nucleolar remodeling complex (NoRC) that regulates the expression of noncoding RNAs. GSK2801 is a selective, cell-permeable inhibitor of the BAZ2 family of bromodomain-containing proteins (IC₅₀s = 9-350 nM in a BAZ2B AlphaScreen). It binds to BAZ2A and BAZ2B with K_d values of 0.26 and 0.14 μM, respectively, and does not interact with the bromodomains of BRD4(BD1), CREBBP, TRIM24/TIF1α, PB1(BD5), PCAF, or ATAD2. See the Structural Genomics Consortium (SGC) website for more information.

Uses

GSK2801 is a selective cell-permeable inhibitor of the BAZ2 (bromodomain-containing protein) interfering with nucleosome spacing during chromatin assembly.

References

[1]. chen p, chaikuad a, bamborough p, et al. discovery and characterization of gsk2801, a selective chemical probe for the bromodomains baz2a and baz2b. journal of medicinal chemistry, 2015.

GSK 2801 Preparation Products And Raw materials

Raw materials

Preparation Products

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GSK 2801 Suppliers

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View Lastest Price from GSK 2801 manufacturers

Career Henan Chemical Co

Product: GSK 2801 1619994-68-1
Price: US $1.00/KG
Min. Order: 1KG
Purity: 95%~99%
Supply Ability: per week 100kg
Release date: 2019-09-05

1619994-68-1, GSK 2801Related Search:

GSK2814338 GSK-2256098 GSK-25 S)-1-(sec-butyl)-N-((4,6-diMethyl-2-oxo-1,2-dihydropyridin-3-yl)Methyl)-3-Methyl-6-(6-(piperazin-1-yl)pyridin-3-yl)-1H-indole-4-carboxaMide 7Methyl-5-(1-{[3-(trifluoroMethyl)phenyl]acetyl}-2,3-dihydro1Hindol-5-yl)7Hpyrrolo[2,3d]pyriMidin-4-aMine GSK2636771 GSK2879552 GSK2795039 GSK 2330672 GSK2838232

GSK 2801

GSK2801

GSK-2801

1-(7-(2-Methylsulfonyl-phenyl)-4-propoxy-1-aza-bicyclo[4.3.0]nona-2,4,6,8-tetraen-9-yl)-ethanone

1-(1-(2-(methylsulfonyl)phenyl)-7-propoxyindolizin-3-yl)ethanone

1-[1-[2-(Methylsulfonyl)phenyl]-7-propoxy-3-indolizinyl]ethanone

GSK2801 GSK-2801

1-[1-(2-Methanesulfonyl-phenyl)-7-propoxy-indolizin-3-yl]-ethanone

GSK2801;GSK-2801;GSK 2801

CS-1607

GSK2801, >98%

GSK 280

GSK-2801; GSK 280

Ethanone, 1-[1-[2-(methylsulfonyl)phenyl]-7-propoxy-3-indolizinyl]-

inhibit,Inhibitor,GSK-2801,TNBC,BAZ2A,GSK2801,Epigenetic Reader Domain,Apoptosis,BAZ2B,cetyl-lysine,orally,GSK 2801

1619994-68-1

Inhibitors