ChemicalBook > CAS DataBase List > GAK inhibitor 49
GAK inhibitor 49
- Product Name
- GAK inhibitor 49
- CAS No.
- 319492-82-5
- Chemical Name
- GAK inhibitor 49
- Synonyms
- AK inhibitor 49;GAK inhibitor 49;GAK inhibitor 49, 10 mM in DMSO;6,7-Dimethoxy-N-(3,4,5-trimethoxyphenyl)quinolin-4-amine;4-Quinolinamine, 6,7-dimethoxy-N-(3,4,5-trimethoxyphenyl)-;NAK,selective,GAK inhibitor-49,GAK inhibitor49,GAK inhibitor 49,Inhibitor,inhibit,ATP-competitive,family
- CBNumber
- CB54667925
- Molecular Formula
- C20H22N2O5
- Formula Weight
- 370.4
- MOL File
- 319492-82-5.mol
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GAK inhibitor 49 Property
- Boiling point:
- 494.8±45.0 °C(Predicted)
- Density
- 1.223±0.06 g/cm3(Predicted)
- storage temp.
- Store at -20°C
- solubility
- DMSO: 50 mg/mL (134.99 mM; ultrasonic and warming and heat to 80°C)
- pka
- 7?+-.0.50(Predicted)
- form
- Solid
- color
- White to off-white
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N-Bromosuccinimide Price
Ambeed
- Product number
- A1359459
- Product name
- 6,7-Dimethoxy-N-(3,4,5-trimethoxyphenyl)quinolin-4-amine
- Purity
- 98%
- Packaging
- 1mg
- Price
- $39
- Updated
- 2021/12/16
Ambeed
- Product number
- A1359459
- Product name
- 6,7-Dimethoxy-N-(3,4,5-trimethoxyphenyl)quinolin-4-amine
- Purity
- 98%
- Packaging
- 5mg
- Price
- $55
- Updated
- 2021/12/16
Ambeed
- Product number
- A1359459
- Product name
- 6,7-Dimethoxy-N-(3,4,5-trimethoxyphenyl)quinolin-4-amine
- Purity
- 98%
- Packaging
- 10mg
- Price
- $100
- Updated
- 2021/12/16
Ambeed
- Product number
- A1359459
- Product name
- 6,7-Dimethoxy-N-(3,4,5-trimethoxyphenyl)quinolin-4-amine
- Purity
- 98%
- Packaging
- 25mg
- Price
- $170
- Updated
- 2021/12/16
Ambeed
- Product number
- A1359459
- Product name
- 6,7-Dimethoxy-N-(3,4,5-trimethoxyphenyl)quinolin-4-amine
- Purity
- 98%
- Packaging
- 50mg
- Price
- $290
- Updated
- 2021/12/16
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GAK inhibitor 49 Chemical Properties,Usage,Production
Uses
GAK inhibitor 49 is a potent, ATP-competitive and highly selective cyclin G associated kinase (GAK) inhibitor with a Ki of 0.54 nM and a cell IC50 of 56 nM. GAK inhibitor 49 also shows binding to RIPK2[1].
References
[1] Asquith CRM, et al. Identification and Optimization of 4-Anilinoquinolines as Inhibitors of Cyclin G Associated Kinase. ChemMedChem. 2018;13(1):48-66. DOI:10.1002/cmdc.201700663
GAK inhibitor 49 Preparation Products And Raw materials
Raw materials
Preparation Products
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GAK inhibitor 49 Suppliers
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