ChemicalBook > CAS DataBase List > L-Alaninamide, N2-acetyl-L-lysyl-L-α-aspartylglycyl-L-isoleucyl-L-valyl-L-asparaginylglycyl-L-valyl-L-lysyl-

L-Alaninamide, N2-acetyl-L-lysyl-L-α-aspartylglycyl-L-isoleucyl-L-valyl-L-asparaginylglycyl-L-valyl-L-lysyl-

Product Name
L-Alaninamide, N2-acetyl-L-lysyl-L-α-aspartylglycyl-L-isoleucyl-L-valyl-L-asparaginylglycyl-L-valyl-L-lysyl-
CAS No.
2243207-00-1
Chemical Name
L-Alaninamide, N2-acetyl-L-lysyl-L-α-aspartylglycyl-L-isoleucyl-L-valyl-L-asparaginylglycyl-L-valyl-L-lysyl-
Synonyms
α-Synuclein 4554W;α-Synuclein Binding?Peptide?trifluoroacetate salt;L-Alaninamide, N2-acetyl-L-lysyl-L-α-aspartylglycyl-L-isoleucyl-L-valyl-L-asparaginylglycyl-L-valyl-L-lysyl-
CBNumber
CB68249388
Molecular Formula
C45H80N14O14
Formula Weight
1041.22
MOL File
2243207-00-1.mol
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L-Alaninamide, N2-acetyl-L-lysyl-L-α-aspartylglycyl-L-isoleucyl-L-valyl-L-asparaginylglycyl-L-valyl-L-lysyl- Property

Boiling point:
1532.8±65.0 °C(Predicted)
Density 
1.241±0.06 g/cm3(Predicted)
pka
4.21±0.10(Predicted)
form 
Solid
color 
White to off-white
Sequence
Ac-Lys-Asp-Gly-Ile-Val-Asn-Gly-Val-Lys-Ala-NH?
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Hazard and Precautionary Statements (GHS)

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L-Alaninamide, N2-acetyl-L-lysyl-L-α-aspartylglycyl-L-isoleucyl-L-valyl-L-asparaginylglycyl-L-valyl-L-lysyl- Chemical Properties,Usage,Production

Uses

α-Synuclein 4554W is an inhibitor of α-Synuclein (aSyn) aggregation with associated toxicity. α-Synuclein 4554W consists of GIVNGVKA sequences, previously identified through intracellular library screening. α-Synuclein 4554W reduces fibril formation of aSyn mutants assocaited with Parkinson’s disease[1].

IC 50

α-synuclein Aggregation

References

[1] Torpey J H, et al. Insights into peptide inhibition of alpha-synuclein aggregation[J]. Frontiers in Neuroscience, 2020, 14: 561462.

L-Alaninamide, N2-acetyl-L-lysyl-L-α-aspartylglycyl-L-isoleucyl-L-valyl-L-asparaginylglycyl-L-valyl-L-lysyl- Preparation Products And Raw materials

Raw materials

Preparation Products

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L-Alaninamide, N2-acetyl-L-lysyl-L-α-aspartylglycyl-L-isoleucyl-L-valyl-L-asparaginylglycyl-L-valyl-L-lysyl- Suppliers

BOC Sciences
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1-631-485-4226; 16314854226
Email
info@bocsci.com
Country
United States
ProdList
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2243207-00-1, L-Alaninamide, N2-acetyl-L-lysyl-L-α-aspartylglycyl-L-isoleucyl-L-valyl-L-asparaginylglycyl-L-valyl-L-lysyl-Related Search:


  • L-Alaninamide, N2-acetyl-L-lysyl-L-α-aspartylglycyl-L-isoleucyl-L-valyl-L-asparaginylglycyl-L-valyl-L-lysyl-
  • α-Synuclein Binding?Peptide?trifluoroacetate salt
  • α-Synuclein 4554W
  • 2243207-00-1
  • C45H80N14O14