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TELENZEPINE DIHYDROCHLORIDE

Product Name
TELENZEPINE DIHYDROCHLORIDE
CAS No.
147416-96-4
Chemical Name
TELENZEPINE DIHYDROCHLORIDE
Synonyms
TelenzepineHydrochloride;Telenzepine dihydrochloide;TELENZEPINE DIHYDROCHLORIDE;JTQJFSQQHGPLOX-UHFFFAOYSA-N;Telenzepine hydrate dihydrochloride;TELENZEPINE DIHYDROCHLORIDE SELECTIVE M1 MUSCARIN;4,9-Dihydro-3-methyl-4-((4-methyl-1-piperazinyl)acetyl)-(10H);4,9-Dihydro-3-methyl-4-((4-methyl-1-piperazinyl)acetyl)-(10H)thieno[3,4-b][1,5]benzodiazepin-10-onedihydrochloride;4,9-DIHYDRO-3-METHYL-4-[(4-METHYL-1-PIPERAZINYL)ACETYL]-10H-THIENO[3,4-B][1,5] BENZODIAZEPIN-10-ONE DIHYDROCHLORIDE
CBNumber
CB8218386
Molecular Formula
C19H22N4O2S
Formula Weight
370.47
MOL File
147416-96-4.mol
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TELENZEPINE DIHYDROCHLORIDE Property

storage temp. 
Store at RT
solubility 
H2O: >10 mg/mL
form 
solid
color 
white
Water Solubility 
Soluble to 100 mM in water
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Safety

WGK Germany 
3
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Hazard and Precautionary Statements (GHS)

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N-Bromosuccinimide Price

Sigma-Aldrich
Product number
T122
Product name
Telenzepine dihydrochloride hydrate
Purity
solid, ≥98% (HPLC)
Packaging
10mg
Price
$80.2
Updated
2024/03/01
Sigma-Aldrich
Product number
T122
Product name
Telenzepine dihydrochloride hydrate
Purity
solid, ≥98% (HPLC)
Packaging
25mg
Price
$129
Updated
2024/03/01
Sigma-Aldrich
Product number
T122
Product name
Telenzepine dihydrochloride hydrate
Purity
solid, ≥98% (HPLC)
Packaging
100mg
Price
$485
Updated
2024/03/01
Tocris
Product number
1122
Product name
Telenzepinedihydrochloride
Purity
≥98%(HPLC)
Packaging
10
Price
$75
Updated
2021/12/16
Tocris
Product number
1122
Product name
Telenzepinedihydrochloride
Purity
≥98%(HPLC)
Packaging
50
Price
$287
Updated
2021/12/16
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TELENZEPINE DIHYDROCHLORIDE Chemical Properties,Usage,Production

Uses

Antiulcerative;M1 muscarinic antagonist

Uses

Telenzepine dihydrochloride is a potent and selective muscarnic receptor antagonist.

Uses

Telenzepine dihydrochloride hydrate was used to study M1 muscarinic receptor-mediated signaling in juvenile rat hippocampus and rat urinary bladder.

Biological Activity

Selective high affinity muscarinic M 1 receptor antagonist (K i = 0.94 nM). Inhibits gastric acid secretion.

Biochem/physiol Actions

Telenzepine is an analog of pirenzepine and inhibits the secretion of gastric acid. It is an antagonist to M1-receptor and targets the oxyntic gastric glands and the salivary glands.

storage

Desiccate at RT

TELENZEPINE DIHYDROCHLORIDE Preparation Products And Raw materials

Raw materials

Preparation Products

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TELENZEPINE DIHYDROCHLORIDE Suppliers

China 15 Germany 3 Switzerland 1 United Kingdom 3 United States 10 Global 32
SIGMA-RBI
Tel
--
Fax
--
Country
Switzerland
ProdList
6896
Advantage
91

147416-96-4, TELENZEPINE DIHYDROCHLORIDERelated Search:

Pirenzepine hydrochloride N1-(2-AMINOPHENYL)-N2,N2-DIMETHYLGLYCINAMIDE N-(2-aminophenyl)-2-(4-methylpiperazin-1-yl)acetamide telenzepine dihydrochloride hydrate PIPERAZINE ACETIC ACID ANILIDE DIHYDROCHLORIDE N-(2-aminophenyl)-2-(diethylamino)acetamide TELENZEPINE DIHYDROCHLORIDE 2-PIPERAZINE-1-YL-ACETAMIDE (PIPERAZIN-1-YL)-ACETAMIDE X 2 HCL X 1/2 H2O

  • 4,9-DIHYDRO-3-METHYL-4-[(4-METHYL-1-PIPERAZINYL)ACETYL]-10H-THIENO[3,4-B][1,5] BENZODIAZEPIN-10-ONE DIHYDROCHLORIDE
  • TELENZEPINE DIHYDROCHLORIDE
  • TELENZEPINE DIHYDROCHLORIDE SELECTIVE M1 MUSCARIN
  • 4,9-Dihydro-3-methyl-4-((4-methyl-1-piperazinyl)acetyl)-(10H)thieno[3,4-b][1,5]benzodiazepin-10-onedihydrochloride
  • Telenzepine dihydrochloide
  • Telenzepine hydrate dihydrochloride
  • 4,9-Dihydro-3-methyl-4-((4-methyl-1-piperazinyl)acetyl)-(10H)
  • JTQJFSQQHGPLOX-UHFFFAOYSA-N
  • TelenzepineHydrochloride
  • 147416-96-4
  • C19H24Cl2N4O2S
  • C19H22N4O2S2HCl
  • C19H22N4O2S
  • Acetylcholine receptor