L-803,087 TRIFLUOROACETATE

Product Name: L-803,087 TRIFLUOROACETATE
CAS No.: 217480-26-7
Chemical Name: L-803,087 TRIFLUOROACETATE
Synonyms: L803087,L 803087;L-803087, 10 mM in DMSO;L-803,087 TRIFLUOROACETATE;Methyl (4-(5,7-difluoro-2-phenyl-1H-indol-3-yl)butanoyl)-L-argininate;L-Arginine, N2-[4-(5,7-difluoro-2-phenyl-1H-indol-3-yl)-1-oxobutyl]-, methyl ester;N2-[4-(5,7-DIFLUORO-2-PHENYL-1H-INDOL-3-YL)-1-OXOBUTYL]-L-ARGININE METHYL ESTER TRIFLUOROACETATE
CBNumber: CB8840994
Molecular Formula: C25H29F2N5O3
Formula Weight: 485.53
MOL File: 217480-26-7.mol

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L-803,087 TRIFLUOROACETATE Property

Density: 1.33±0.1 g/cm3(Predicted)
storage temp.: Store at -20°C
solubility: Soluble to 100 mM in DMSO and to 100 mM in ethanol
form: Powder
pka: 14.54±0.46(Predicted)
color: White to light yellow

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Hazard and Precautionary Statements (GHS)

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N-Bromosuccinimide Price

Tocris

Product number: 1979
Product name: L-803,087trifluoroacetate
Purity: ≥97%(HPLC)
Packaging: 10
Price: $331
Updated: 2021/12/16

TRC

Product number: L011600
Product name: L803087
Packaging: 2.5mg
Price: $310
Updated: 2021/12/16

Usbiological

Product number: 255643
Product name: L-803,087 trifluoroacetate
Packaging: 10mg
Price: $588
Updated: 2021/12/16

ChemScene

Product number: CS-0028987
Product name: L-803087
Purity: >98.0%
Packaging: 5mg
Price: $650
Updated: 2021/12/16

ChemScene

Product number: CS-0028987
Product name: L-803087
Purity: >98.0%
Packaging: 1mg
Price: $250
Updated: 2021/12/16

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L-803,087 TRIFLUOROACETATE Chemical Properties,Usage,Production

Uses

Somatostatin receptors are often overexpressed in tumours and are potential therapeutic targets. Somatostatin receptor agonists can be used to study signaling pathways related somatostatin receptor. L 803087 is a somatostatin sst4 receptor agonist.

Biological Activity

Potent and selective somatostatin sst 4 receptor agonist. K i values are 0.7, 199, 4720, 1280 and 3880 nM for cloned human sst 4 , sst 1 , sst 2 , sst 3 and sst 5 receptors respectively. Facilitates AMPA-mediated hippocampal synaptic responses in vitro and increases kainate-induced seizures in mice in vivo .

in vivo

L-803087 (5 nmol) is doubled seizure activity in wild-type mice on average. Interestingly, this effect is blocked by 3 nmol Octreotide. In hippocampal slices from wild-type mice, Octreotide (2 μM) does not modify AMPA-mediated synaptic responses while facilitation occurred with L-803087 (2 μM)^[2].

L-803,087 TRIFLUOROACETATE Preparation Products And Raw materials

Raw materials

Preparation Products

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L-803,087 TRIFLUOROACETATE Suppliers

China 22 Europe 1 Germany 3 United Kingdom 1 United States 6 Global 33

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217480-26-7, L-803,087 TRIFLUOROACETATERelated Search:

CDH Dodecyl acrylate L-803,087 TRIFLUOROACETATE

N2-[4-(5,7-DIFLUORO-2-PHENYL-1H-INDOL-3-YL)-1-OXOBUTYL]-L-ARGININE METHYL ESTER TRIFLUOROACETATE

L-803,087 TRIFLUOROACETATE

L-Arginine, N2-[4-(5,7-difluoro-2-phenyl-1H-indol-3-yl)-1-oxobutyl]-, methyl ester

L803087,L 803087

Methyl (4-(5,7-difluoro-2-phenyl-1H-indol-3-yl)butanoyl)-L-argininate

L-803087, 10 mM in DMSO

217480-26-7

C25H29F2N5O3CF3CO2H

C25H29F2N5O3

Somatostatin receptor