1-BOC-INDOLE Chemical Properties

Melting point:

24-26

Boiling point:

201 °C(lit.)

Density 

1.07 g/mL at 25 °C(lit.)

refractive index 

n20/D 1.543(lit.)

Flash point:

160 °F

storage temp. 

Sealed in dry,2-8°C

form 

liquid

Specific Gravity

1.070

color 

Yellow

BRN 

4674239

CAS DataBase Reference

75400-67-8(CAS DataBase Reference)

Safety Information

Hazard Codes 

Xi

Safety Statements 

24/25

WGK Germany 

3

Hazard Note 

Irritant/Keep Cold

HazardClass 

IRRITANT, KEEP COLD

HS Code 

2933998090

MSDS

• Language:English Provider:SigmaAldrich
• Language:English Provider:ALFA

1-BOC-INDOLE Usage And Synthesis

Uses

Reactant for preparation of:

• Potent plant-growth inhibitors
• Cannabinoid CB2 receptor ligands
• Analogues of isomeridianin G and evaluation as GSK-3β inhibitors
• Inhibitor of the Yersinia pestis salicylate adenylation domain YbtE
• Cholecystokinin-2 receptor antagonists
• Antileishmanial agents

• Reactant for:
• Palladium-catalyzed Suzuki-Miyaura cross coupling reactions
• Friedel-Crafts alkylation reactions

Synthesis Reference(s)

Tetrahedron Letters, 43, p. 4115, 2002 DOI: 10.1016/S0040-4039(02)00696-2

1-BOC-INDOLE(75400-67-8)Related Product Information

• tert-butyl 1-ethylhydrazine-1-carboxylate
• tert-butyl 2-(2-oxoiMidazolidin-1-yl)acetate
• tert-butyl 2-(3-benzoylthioureido)-5,5-diMethyl-5,7-dihydro-4H-thieno[2,3-c]pyran-3-carboxylate
• N-BOC-INDOLE-2-BORONIC ACID,1-(N-BOC)-INDOLE-2-BORONIC ACID,1-BOC-INDOLE-2-BORONIC ACID
• 1-BOC-INDOLE
• BOC-TRP(BOC)-OH
• 5-BENZYLOXY-1-BOC-INDOLE-2-BORONIC ACID
• 5-BROMO-N-(BOC)INDOLE-2-BORONIC ACID
• 6-BENZYLOXY-1-BOC-INDOLE-2-BORONIC ACID
• 4-CHLORO-N-(BOC)-INDOLE-2-BORONIC ACID
• 4-BENZYLOXY-1-BOC-INDOLE-2-BORONIC ACID
• Fmoc-Trp(Boc)-OH
• TERT-BUTYL 5-BROMOINDOLE-1-CARBOXYLATE
• N-Boc-2-pyrroleboronic acid
• Fmoc-D-Trp(Boc)-OH
• Z-TRP(BOC)-OH DCHA
• H-TRP(BOC)-OH
• FMOC-METRP(BOC)-OH