Basic information Safety Supplier Related

(S)-Maleoyl-DPR(Boc)-OH·DCHA

Basic information Safety Supplier Related

(S)-Maleoyl-DPR(Boc)-OH·DCHA Basic information

Product Name:
(S)-Maleoyl-DPR(Boc)-OH·DCHA
Synonyms:
  • (S)-Maleoyl-DPR(Boc)-OH·DCHA
  • Mal-Dap(Boc)·DCHA
  • Mal-Dpr(Boc)·DCHA
  • Mal-L-Dap(Boc)-OH·DCHA≥99%
  • Mal-L-PA-NH-Boc
  • mDPR(boc)
  • 1H-Pyrrole-1-acetic acid, α-[[[(1,1-dimethylethoxy)carbonyl]amino]methyl]-2,5-dihydro-2,5-dioxo-, (αS)-
  • (S)-3-((tert-Butoxycarbonyl)amino)-2-(2,5-dioxo-2,5-dihydro-1H-pyrrol-1-yl)propanoic acid
CAS:
1491152-23-8
MF:
C12H16N2O6
MW:
284.27
Mol File:
1491152-23-8.mol
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(S)-Maleoyl-DPR(Boc)-OH·DCHA Chemical Properties

Boiling point:
494.4±40.0 °C(Predicted)
Density 
1.368±0.06 g/cm3(Predicted)
pka
3.03±0.10(Predicted)
form 
Solid
color 
White to off-white
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(S)-Maleoyl-DPR(Boc)-OH·DCHA Usage And Synthesis

Uses

Mal-L-PA-NH-Boc is a noncleavable ADC linker used in the synthesis of antibody-drug conjugates (ADCs).

IC 50

Non-cleavable Linker

References

[1] Robert Lyon, et al. Self-stabilizing linker conjugates. WO2013173337A2.

(S)-Maleoyl-DPR(Boc)-OH·DCHASupplier

Accela ChemBio Co.,Ltd.
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021-50795510 4000665055
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sales@accelachem.com
Zhongshan Resi Biotechnology Co., Ltd.
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13715524166 13326948089
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resicn@resicn.com
Jinan Kabotang Biological Technology Co.,Ltd.
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0531-61320525 15866703830
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figo.gao@foxmail.com
Fan De(Beijing) Biotechnology Co., Ltd.
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15911056312
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liming@bio-fount.com
TargetMol Chemicals Inc.
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+1-781-999-5354; +17819995354
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marketing@targetmol.com