Basic information Safety Supplier Related

Almitrine dimesylate

Basic information Safety Supplier Related

Almitrine dimesylate Basic information

Product Name:
Almitrine dimesylate
Synonyms:
  • ALMITRINE BISMESYLATE
  • ALMITRINE DIMESYLATE
  • 2,4-bis(allylamino)-6-[4-[bis(p-fluorophenyl)methyl]-1-piperazinyl]-s-triazine dimethanesulfonate
  • n,n'-diallyl-6-[4-[bis(4-fluorophenyl)methyl]piperazin-1-yl]-1,3,5-triazine-2,4-diamine dimethanesulphonate
  • ALMITRINE DIMESILATE
  • Mesylate AlMitrine
  • N2,N4-Diallyl-6-(4-(bis(4-fluorophenyl)methyl)piperazin-1-yl)-1,3,5-triazine-2,4-diamine dimethanesulfonate
  • Almitrine bismethanesulfonate
CAS:
29608-49-9
MF:
C28H37F2N7O6S2
MW:
669.76
EINECS:
249-726-1
Product Categories:
  • API
Mol File:
29608-49-9.mol
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Almitrine dimesylate Chemical Properties

Melting point:
243° (dec)
storage temp. 
Sealed in dry,Room Temperature
solubility 
Chloroform (Slightly), Methanol (Slightly)
form 
Solid
color 
White
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Safety Information

Toxicity
LD50 in mice: 210 mg/kg i.v., 390 mg/kg i.p., >2 g/kg orally (Regnier)
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Almitrine dimesylate Usage And Synthesis

Uses

Respiratory stimulant.

Definition

ChEBI: The dimethanesulfonate salt of almitrine.

brand name

Vectarion (Oril S.A., France).

in vivo

Almitrine acts via the peripheral arterial chemoreceptors raising carotid sinus nerve output and minute ventilation. Almitrine also has a pulmonary vascular action causing a dose-dependent constriction and dilatation. At low doses Almitrine enhances hypoxic pulmonary vasoconstriction and may improve the overall ventilation/perfusion ratio[2].

Almitrine dimesylateSupplier

Dalian Meilun Biotech Co., Ltd.
Tel
0411-62910999 13889544652
Email
sales@meilune.com
Guangzhou Isun Pharmaceutical Co., Ltd
Tel
020-39119399 18927568969
Email
isunpharm@qq.com
Bide Pharmatech Ltd.
Tel
400-164-7117 13681763483
Email
product02@bidepharm.com
Wuhan Dahua Pharmaceutical Co., Ltd.
Tel
027-59262863 13277907145 3091977954
Shanghai QianJin Chemical Technology Co., Ltd
Tel
021-20900665 17321230821
Email
2986274987@qq.com