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PAROXETINE-D4 HCL

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PAROXETINE-D4 HCL Basic information

Product Name:
PAROXETINE-D4 HCL
Synonyms:
  • Piperidine, 3-[(1,3-benzodioxol-5-yloxy)methyl]-4-(4-fluorophenyl)-, hydrochloride, hydrate (2:1), (3S,4R)- (9CI)
  • 1,3-benzodioxol-5-yl-[4-(4-fluorophenyl)-3-piperidinyl]methanol hydrochloride
  • PAROXETINE-D4 HCL kf-yuwen(at)kf-chem.com
  • Piperidine, 3-[(1,3-benzodioxol-5-yloxy)methyl]-4-(4-fluorophenyl)-, hydrochloride, hydrate (2:1), (3S-trans)-
  • Paroxetine Hydrochloride (350 mg)
  • Paroxetine Hydrochloride (350 mg)G0D0030.972mg/mg(ai)
  • Paroxetine-D4 hydrochloride
  • PAROXETINE-D4 HCL
CAS:
110429-35-1
MF:
C19H23ClFNO4
MW:
383.84
EINECS:
000-000-0
Product Categories:
  • Active Pharmaceutical Ingredients
  • Cnbio
  • Serotonin
Mol File:
110429-35-1.mol
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PAROXETINE-D4 HCL Chemical Properties

Melting point:
121-131 C
storage temp. 
under inert gas (nitrogen or Argon) at 2-8°C
solubility 
Slightly soluble in water, freely soluble in methanol, sparingly soluble in ethanol (96 per cent) and in methylene chloride.
form 
powder
color 
white
λmax
292nm(H2O)(lit.)
Merck 
14,7043
CAS DataBase Reference
110429-35-1
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Safety Information

Hazard Codes 
F,C,Xn
Risk Statements 
11-34-36/37/38-22
Safety Statements 
16-26-36/37/39-45-36
RIDADR 
UN 3077 9 / PGIII
WGK Germany 
3
RTECS 
TM4569320
HazardClass 
IRRITANT
HS Code 
29349990
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PAROXETINE-D4 HCL Usage And Synthesis

Chemical Properties

White or almost white, crystalline powder.

Uses

Paroxetine Hydrochloride, is a selective serotonin reuptake inhibitor (SSRI) antidepressant used to treat depression, panic attacks, obsessive-compulsive disorder (OCD), anxiety disorders, post-traumatic stress disorder, and a severe form of premenstrual syndrome (premenstrual dysphoric disorder).

Uses

Antidepressant;5-HT uptake inhibitor

Uses

Paroxetine hydrochloride hemihydrate has been used: as an antidepressant to study its effects on neural stem cells (NSCs) from embryonic rat hippocampus in vitro; as a CYP 2D6 inhibitor to study its effects on the in vitro?production by human recombinant CYP 2D6 of the phenolic metabolites; as an antidepressant to study its effects on the expression of pituitary adenylate cyclase activating polypeptide (PACAP), its receptors and brain-derived neurotrophic factor (BDNF) in rat primary hippocampal neurons

General Description

Pharmaceutical secondary standards for application in quality control provide pharma laboratories and manufacturers with a convenient and cost-effective alternative to the preparation of in-house working standards

Biochem/physiol Actions

Paroxetine hydrochloride hemihydrate is one of the most potent and selective of the selective serotonin reuptake inhibitors (SSRI); antidepressant

in vivo

Paroxetine treatment obviously attenuates the symptoms of CIA rats. Paroxetine treatment clearly prevents the histological damage of joints and alleviates T cells infiltration into synovial tissue. Paroxetine reveals a strong effect on inhibiting CX3CL1 production in synovial tissues[1]. Paroxetine (20 mg/kg/day) reduces the myocyte cross-sectional area in rat and ROS formation in the remote myocardium. Paroxetine reduces the susceptibility to ventricular tachycardia. Paroxetine treatment following MI decreases LV remodeling and susceptibility to arrhythmias, probably by reducing ROS formation[2]. In CCI paroxetine-treated group, paroxetine (10 mg/kg, i.p.) produces hyperalgesia at days 7 and 10 (P<0.01), but a decrease in pain behavior is seen at day 14. Moreover, paroxetine (10 mg/kg) significantly attenuates tactile hypersensitivity when compared to CCI vehicle-treated group[5].

PAROXETINE-D4 HCL Preparation Products And Raw materials

Preparation Products

PAROXETINE-D4 HCLSupplier

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