LY-2608204
LY-2608204 Basic information
- Product Name:
- LY-2608204
- Synonyms:
-
- LY-2608204
- (1R,2S)-2-Cyclohexyl-1-[4-(cyclopropylsulfonyl)phenyl]-N-[5-[[2-(1-pyrrolidinyl)ethyl]thio]-2-thiazolyl]cyclopropanecarboxamide
- (1R,2S)-2-cyclohexyl-1-(4-(cyclopropylsulfonyl)phenyl)-N-(5-((2-(pyrrolidin-1-yl)ethyl)thio)thiazol-2-yl)cyclopropanecarboxaMide
- CS-898
- LY-2608204; LY 2608204
- (1R,2S)-2-Cyclohexyl-1-[4-(cyclopropylsulfonyl)phenyl]-N-[5-[[2-(1-pyrrolidinyl)ethyl]thio]-2-thiazolyl]cyclopropanecarboxamide LY 2608204
- Cyclopropanecarboxamide, 2-cyclohexyl-1-[4-(cyclopropylsulfonyl)phenyl]-N-[5-[[2-(1-pyrrolidinyl)ethyl]thio]-2-thiazolyl]-, (1R,2S)-
- LY-2608024
- CAS:
- 1234703-40-2
- MF:
- C28H37N3O3S3
- MW:
- 559.81
- Product Categories:
-
- Inhibitors
- Mol File:
- 1234703-40-2.mol
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LY-2608204 Chemical Properties
- Density
- 1.35
- storage temp.
- Store at -20°C
- solubility
- ≥28.35 mg/mL in DMSO; insoluble in H2O; ≥26.2 mg/mL in EtOH
- form
- solid
- pka
- 8.17±0.70(Predicted)
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LY-2608204 Usage And Synthesis
Description
LY2608204 is an activator of glucokinase (GK; EC50 = 42 nM). It stimulates glucose metabolism in INS-1E rat insulinoma cells (mean EC50 = 579 nM). LY2608204 (30 mg/kg) decreases plasma glucose levels in a dose-dependent manner in fasted rats.
target
GK
References
[1] kj filipski, bd stevens . glucokinase activators in development .2012 books
LY-2608204Supplier
Shanghai Boyle Chemical Co., Ltd.
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- sales@boylechem.com
Dalian Meilun Biotech Co., Ltd.
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- 0411-62910999 13889544652
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Haoyuan Chemexpress Co., Ltd.
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- 021-58950125
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Shanghai Aladdin Bio-Chem Technology Co.,LTD
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- 400-6206333 18521732826;
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shanghai cooperpharm co.,LTD .
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- +86-021-58975553
- sales@cooperpharm.com