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Pentoxyverine

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Pentoxyverine Basic information

Product Name:
Pentoxyverine
Synonyms:
  • 1-phenyl-1-cyclopentanecarboxylic acid 2-[2-(diethylamino)ethoxy]ethyl ester
  • 1-phenyl-1-cyclopentanecarboxylate
  • 1-Phenylcyclopentane-1-Carboxylic acid diethylaminoethoxyethyl ester
  • 1-phenylcyclopentane-1-carboxylicaciddiethylaminoethoxyethylester
  • 1-phenyl-cyclopentanecarboxylicaci2-(2-(diethylamino)ethoxy)ethylester
  • 1-phenylcyclopentanecarboxylicacid2-(2-diethylaminoethoxy)ethylester
  • ucb2543
  • Urex
CAS:
77-23-6
MF:
C20H31NO3
MW:
333.46
EINECS:
201-014-1
Product Categories:
  • Miscellaneous Biochemicals
Mol File:
77-23-6.mol
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Pentoxyverine Chemical Properties

Boiling point:
165-170 °C (1.33Pa)
Density 
1.048±0.06 g/cm3(Predicted)
refractive index 
1.4990-1.5010
storage temp. 
Refrigerator
solubility 
Dichloromethane (Slightly), Methanol (Slightly)
pka
9.69±0.25(Predicted)
form 
Oil
color 
Clear Very Dark Red to Brown
CAS DataBase Reference
77-23-6(CAS DataBase Reference)
NIST Chemistry Reference
1-Cyclopentanecarboxylate, 2-(diethylaminoethoxy)ethyl-1-phenyl-(77-23-6)
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Safety Information

Hazardous Substances Data
77-23-6(Hazardous Substances Data)
Toxicity
LD50 oral in rat: 150mg/kg
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Pentoxyverine Usage And Synthesis

Originator

Asthma ,Nichiiko

Uses

Carbetapentane is an antitussive anticonvulsant sigma site agonist.

Definition

ChEBI: 1-phenyl-1-cyclopentanecarboxylic acid 2-[2-(diethylamino)ethoxy]ethyl ester is a member of benzenes.

Manufacturing Process

1-Phenylcyclopentane carbonitrile was obtained by treatment of phenylacetonitrile with sodium amide and 1,4-dibrombutane.
1-Phenyl-1-cyclopentane carboxylic acid was produced in the result of reaction of 1-phenylcyclopentane carbonitrile with sulfuric acid.
1-Phenyl-1-cyclopentanecarbonyl chloride was obtained by treatment of 1phenyl-1-cyclopentane carboxylic acid with thionyl chloride.
A mixture of 0.5 mol of 1-phenyl-1-cyclopentanecarbonyl chloride and of 0.5 mol of 2-(2-diethylaminoethoxy)ethanol (herein-after referred to as the amino alcohol) in 300 ml of toluene is heated under reflux for 20 h. The mixture is thereafter made alkaline by means of an aqueous solution of caustic soda and decanted; the toluenic layer is washed with water and concentrated in vacuo. The residue is distilled under high vacuum. After two fractional distillations, the 2-(2-diethylaminoethoxy)ethyl 1-phenylcyclopentane-carboxylate is obtained, in 85% yield. Boiling point 164°C/0.1 mm. Hg.

brand name

Toclase (Pfizer).

Therapeutic Function

Antitussive

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