PIBOSEROD,2H-(1,3)OXAZINO(3,2-A)INDOLE-10-CARBOXAMIDE, N-((1-BUTYL-4-PIPERIDINYL)METHYL)-3,4-DIHYDRO- Chemical Properties

Melting point:

110-113°

Boiling point:

570.3±35.0 °C(Predicted)

Density 

1.22±0.1 g/cm3(Predicted)

storage temp. 

2-8°C

solubility 

DMF: 30 mg/mL; DMSO: 20 mg/mL; Ethanol: 30 mg/mL; Ethanol:PBS (pH7.2)(1:20): 0.05 mg/mL

pka

13.86±0.20(Predicted)

form 

powder

color 

white to beige

Safety Information

RIDADR 

UN 2811 6.1 / PGIII

PIBOSEROD,2H-(1,3)OXAZINO(3,2-A)INDOLE-10-CARBOXAMIDE, N-((1-BUTYL-4-PIPERIDINYL)METHYL)-3,4-DIHYDRO- Usage And Synthesis

Uses

Treatment of irritable bowel syndrome (selective 5HT4receptor antagonist).

Uses

Piboserod is a 5-HT4 receptor antagonist which has shown positive results as a Hepatitis C virus (HCV) entry inhibtor.

Biochem/physiol Actions

SB-207266 is a potent, selective, orally active and long-acting 5-HT4 antagonist in vivo.

PIBOSEROD,2H-(1,3)OXAZINO(3,2-A)INDOLE-10-CARBOXAMIDE, N-((1-BUTYL-4-PIPERIDINYL)METHYL)-3,4-DIHYDRO-(152811-62-6)Related Product Information

• PIBOSEROD,2H-(1,3)OXAZINO(3,2-A)INDOLE-10-CARBOXAMIDE, N-((1-BUTYL-4-PIPERIDINYL)METHYL)-3,4-DIHYDRO-
• 4-Acetylaminomethyl Piperidine
• (1-Methyl-1H-indol-3-yl)-methylamine
• 1H-Indole-3-carboxamide(9CI)
• 1H-indol-2-ol
• 1-METHYL-1H-INDOL-2-OL