Basic information Safety Supplier Related

NALTRIBEN MESYLATE

Basic information Safety Supplier Related

NALTRIBEN MESYLATE Basic information

Product Name:
NALTRIBEN MESYLATE
Synonyms:
  • NTB
  • NALTRIBEN MESYLATE
  • NALTRIBEN METHANESULFONATE
  • naltrindolebenzofuran
  • 17-(Cyclopropylmethyl)-6,7-didehydro-3-4,5alpha-epoxy-14beta-dihydroxy-6,7-2',3'-benzo[b]furanomorphinan mesylate
  • 17-(Cyclopropylmethyl)-6,7-didehydro-3,14β-dihydroxy-4,5α-epoxy-6,7-2',3'-benzo[b]furanomorphinanmesylate
  • 17-(CYCLOPROPYLMETHYL)-6,7-DIDEHYDRO-3, 14B-DIHYDROXY-4,5A-EPOXY-6,7-2',3'-BENZO[B]FURANOMORPHINAN MESYLATE
  • 17-(Cyclopropylmethyl)-6,7-didehydro-3,14b-dihydroxy-4,5a-epoxy-6,7-2',3'-benzo[b]furanomorphinanmesylate
CAS:
111555-58-9
MF:
C26H25NO4
MW:
415.48
Product Categories:
  • Opioid receptor and opioid-like receptor
Mol File:
111555-58-9.mol
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NALTRIBEN MESYLATE Chemical Properties

Boiling point:
605.3±55.0 °C(Predicted)
Density 
1.50±0.1 g/cm3(Predicted)
storage temp. 
−20°C
solubility 
DMSO: 14 mg/mL at ~60 °C
form 
solid
pka
9.30±0.40(Predicted)
color 
off-white
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Safety Information

WGK Germany 
3
RTECS 
PB9175000
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NALTRIBEN MESYLATE Usage And Synthesis

Uses

Naltriben is a potent and selective antagonist for the δ2 opioid receptor. Naltriben is used to differentiate the δ1 and δ2 opioid receptors.

Definition

ChEBI: Naltriben is a morphinane alkaloid.

Biological Activity

Selective and potent δ -opioid receptor antagonist (K i values are 0.013, 19 and 152 nM for δ , μ and κ receptors respectively). Displays selectivity for the δ 2 subtype in vivo .

NALTRIBEN MESYLATESupplier

3B Pharmachem (Wuhan) International Co.,Ltd.
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821-50328103-801 18930552037
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3bsc@sina.com
EMMX Biotechnology LLC
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888-539-0666
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info@emmx.com
Shanghai Universal Biotech Co.,Ltd
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15921930842 15921930842
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zhouzz@univ-bio.com
Carbosynth
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