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Succinylsulfathiazole

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Succinylsulfathiazole Basic information

Product Name:
Succinylsulfathiazole
Synonyms:
  • colistatin
  • cremosuxidine
  • kaoxidin
  • KAOXIDINE
  • sulfasuccidin
  • sulfasuccidine
  • sulfasuccinil
  • sulfasuccithiazole
CAS:
116-43-8
MF:
C13H13N3O5S2
MW:
355.39
EINECS:
204-141-0
Product Categories:
  • SULFASUXIDINE
  • Antibacterial
  • Antibiotics
  • Antibiotics A to
  • Antibiotics N-SAntibiotics
  • Chemical Structure Class
  • Antibiotics for Research and Experimental Use
  • Biochemistry
  • Sulfonamides (Antibiotics for Research and Experimental Use)
  • Inhibits an EnzymeAntibiotics
  • Interferes with DNA SynthesisSpectrum of Activity
  • L - ZAntibiotics
  • Mechanism of Action
  • Sulfonamides
Mol File:
116-43-8.mol
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Succinylsulfathiazole Chemical Properties

Melting point:
193.5°C
Density 
1.4807 (rough estimate)
refractive index 
1.6390 (estimate)
storage temp. 
Sealed in dry,Room Temperature
solubility 
1 M NaOH: soluble50mg/mL
pka
pKa 4.5 (Uncertain)
form 
powder
color 
white to off-white
Water Solubility 
0.49g/L(38 ºC)
λmax
282nm(H2O (pH 3.3 - 5))(lit.)
Merck 
14,8877
BRN 
349989
CAS DataBase Reference
116-43-8(CAS DataBase Reference)
EPA Substance Registry System
Butanoic acid, 4-oxo-4-[[4-[(2-thiazolylamino)sulfonyl]phenyl]amino]- (116-43-8)
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Safety Information

Hazard Codes 
Xn
Risk Statements 
42/43
Safety Statements 
22-36/37-45
RIDADR 
3249
WGK Germany 
3
RTECS 
WM4767000
HazardClass 
6.1(b)
PackingGroup 
III
HS Code 
29350090

MSDS

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Succinylsulfathiazole Usage And Synthesis

Originator

Sulfasuxidine,MSD,US,1942

Uses

Succinylsulfathiazole is a sulfonamide antibiotic that was shown to inhibit bacteria that are responsible for folate production. Succinylsulfathiazole was used in various folate deficiency studies to block the synthesis of folic acid.

Uses

Succinylsulfathiazole is antibacterial

Definition

ChEBI: N-succinylsulfathiazole is a member of 1,3-thiazoles. It is functionally related to a sulfathiazole.

Manufacturing Process

3.92 g of succinic anhydride was added to a boiling suspension of 10 g of 2- sulfanilamidothiazole in 100 cc of alcohol. The mixture was then refluxed for five minutes after the addition was complete at which time all of the solids were in solution. The solution was then cooled and diluted with an equal volume of water. The white solid precipitate which formed was filtered and recrystallized from dilute alcohol, yielding 2-N4-succinylsulfanilamidothiazole, melting at 184°C to 186°C.

Therapeutic Function

Antibacterial (intestinal)

SuccinylsulfathiazoleSupplier

Creasyn Finechem(Tianjin) Co., Ltd.
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022-83946278 13820503911
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J & K SCIENTIFIC LTD.
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Meryer (Shanghai) Chemical Technology Co., Ltd.
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3B Pharmachem (Wuhan) International Co.,Ltd.
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TCI (Shanghai) Development Co., Ltd.
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021-67121386
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