Basic information Safety Supplier Related

LIDORESTAT

Basic information Safety Supplier Related

LIDORESTAT Basic information

Product Name:
LIDORESTAT
Synonyms:
  • LIDORESTAT
  • 1H-Indole-1-aceticacid, 3-[(4,5,7-trifluoro-2-benzothiazolyl)methyl]-
  • 2-(3-((4,5,7-TRIFLUOROBENZO[D]THIAZOL-2-YL)METHYL)-1H-INDOL-1-YL)ACETIC ACID
  • [3-(4,5,7-Trifluorobenzothiazol-2-ylmethyl)indol-1-yl]acetic acid
  • 3-[(4,5,7-Trifluorobenzothiazol-2-yl)methyl]indole-N-acetic acid
  • LIDORESTATUM
  • IDD-676
  • (VOI)LIDORESTAT
CAS:
245116-90-9
MF:
C18H11F3N2O2S
MW:
376.35
Mol File:
245116-90-9.mol
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LIDORESTAT Chemical Properties

Melting point:
177-178℃
Boiling point:
591.4±50.0 °C(Predicted)
Density 
1.55
form 
Solid
pka
4.23±0.10(Predicted)
color 
Light yellow to yellow
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LIDORESTAT Usage And Synthesis

Uses

Treat ment of diabetic complications, including neuropathy, retinopathy, cataracts, nephropathy (selective aldose reductase inhibitor).

in vivo

Lidorestat (25 mg/kg/day; oral administration; twice daily; for 6 weeks; diabetic mice) treatment decreases fructose and reduces mortality in diabetic hAR-expressing mice. And Lidorestat does not affect weight[1].

Animal Model:Diabetic low-density lipoprotein (LDL) receptor-deficient [Ldlr(-/-)] mice[1]
Dosage:25 mg/kg/day
Administration:Oral administration; twice daily; for 6 weeks
Result: Diabetic hAR-expressing mice had decreased fructose and reduced mortality.

LIDORESTATSupplier

Cochemical Ltd.
Tel
029-86115547 17791676824
Email
sales@cochemical.com
Wuxi AppTec
Tel
022-59987777 13552403979
Email
jia_guoqiang@wuxiapptec.com
Aikon International Limited
Tel
025-58859352 18068836627
Email
dt3@aikonchem.com
3A Chemicals
Tel
400-668-9898
Email
service@3achem.com
Shanghai Jizhi Biochemical Technology Co. Ltd.
Tel
4009004166/18616739031 18616739031
Email
3007523370@qq.com
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LIDORESTAT(245116-90-9)Related Product Information