S(-)-WIN 55 212-3 MESYLATE
S(-)-WIN 55 212-3 MESYLATE Basic information
- Product Name:
- S(-)-WIN 55 212-3 MESYLATE
- Synonyms:
-
- [(3S)-2,3-DIHYDRO-5-METHYL-3-(4-MORPHOLINYLMETHYL)PYRROLO[1,2,3-DE]-1,4-BENZOXAZIN-6-YL]-1-NAPHTHALENYL-METHANONE MONOMETHANESULFONATE
- WIN 55,212-3 MESYLATE
- S(-)-[2,3-Dihydro-5-methyl-3-[(4-morpholinyl)methyl]pyrrolo[1,2,3-de]-1,4-benzoxazinyl]-(1-naphthalenyl)methanone mesylate salt
- S(-)-WIN 55,212-3 mesylate salt
- [(3S)-2,3-Dihydro-5-methyl-3-(4-morpholinylmethyl)pyrrolo[1,2,3-de]-1,4-benzoxazin-6-yl]-1-naphthalenyl-methanonemonomethanesulfonate
- FSGCSTPOPBJYSX-BDQAORGHSA-N
- Methanone, [(3S)-2,3-dihydro-5-methyl-3-(4-morpholinylmethyl)pyrrolo[1,2,3-de]-1,4-benzoxazin-6-yl]-1-naphthalenyl-, methanesulfonate (1:1)
- CAS:
- 131543-25-4
- MF:
- C28H30N2O6S
- MW:
- 522.6126
- Mol File:
- 131543-25-4.mol
More
Less
S(-)-WIN 55 212-3 MESYLATE Chemical Properties
- storage temp.
- Store at +4°C
- solubility
- 45% (w/v) aq 2-hydroxypropyl-β-cyclodextrin: 2.4 mg/mL
- form
- solid
- color
- off-white
More
Less
S(-)-WIN 55 212-3 MESYLATE Usage And Synthesis
Uses
WIN 552,12-3 Mesylate is a high affinity cannabinoid agonist.
Biological Activity
Novel, low potency CB 2 receptor silent antagonist and CB 1 receptor partial inverse agonist. Competitively antagonizes effects of CP 55,940 (pA 2 = 6.1) and SR 144528 (pEC 50 = 5.3) at CB 2 receptors and acts as a partial inverse agonist at CB 1 receptors (pIC 50 = 5.5). Displays modest activity at human melatonin MT 1 and muscarinic M 4 receptors, but is selective over several other GPCRs.
S(-)-WIN 55 212-3 MESYLATESupplier
3B Pharmachem (Wuhan) International Co.,Ltd.
- Tel
- 821-50328103-801 18930552037
- 3bsc@sina.com
EMMX Biotechnology LLC
- Tel
- 888-539-0666
- info@emmx.com
ChemeGen(Shanghai) Biotechnology Co.,Ltd.
- Tel
- 18818260767
- sales@chemegen.com
Nanjing Tengyi Biotechnology Co., Ltd
- Tel
- 025-58851786 17714337195
- sales@tybiochem.com
Shanghai Yifei Biotechnology Co. , Ltd.
- Tel
- 021-65675885 18964387627
- customer_service@efebio.com
More
Less
S(-)-WIN 55 212-3 MESYLATE(131543-25-4)Related Product Information
- 3-benzoylindole
- 1H-Indole-3-carboxaldehyde,2-methyl-1-(1-methylethyl)-(9CI)
- 1-(1-ETHYL-1H-INDOL-3-YL)ETHANONE
- [1-[2-(4-Morpholinyl)ethyl]-1H-indol-3-yl]-1-naphthalenylmethanone
- ASISCHEM W99822
- 3-BENZYLINDOLE
- 1-ISOPROPYL-1H-INDOLE-3-CARBALDEHYDE
- 4-(2-aminopropyl)morpholine
- 1-ETHYL-1H-INDOLE-3-CARBALDEHYDE
- 2-(1H-INDOL-1-YL)ETHANAMINE
- 2-(2-METHYL-1H-INDOL-1-YL)ETHANAMINE
- 7-Methoxy-1H-indole
- 7-Methoxy-3-indolecarboxaldehyde
- 7-Hydroxyindole
- S(-)-WIN 55 212-3 MESYLATE