Basic information Safety Supplier Related

GSK-2881078

Basic information Safety Supplier Related

GSK-2881078 Basic information

Product Name:
GSK-2881078
Synonyms:
  • GSK2881078; GSK 2881078
  • SARM GS2881078
  • CS-2336
  • GSK-2881078
  • GSK-2881078 (Free base)
  • 1H-Indole-5-carbonitrile, 1-[(1R)-1-methyl-2-(methylsulfonyl)ethyl]-4-(trifluoromethyl)-
  • 1-[(2R)-1-(Methylsulfonyl)-2-propanyl]-4-(trifluoromethyl)-1H-indole-5-carbonitrile
  • 1-(1-Methylsulfonylpropan-2-yl)-4-(trifluoromethyl)indole-5-carbonitrile
CAS:
1539314-06-1
MF:
C14H13F3N2O2S
MW:
330.33
EINECS:
1539314-060-1
Mol File:
1539314-06-1.mol
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GSK-2881078 Chemical Properties

Boiling point:
521.6±50.0 °C(Predicted)
Density 
1.36±0.1 g/cm3(Predicted)
storage temp. 
Store at -20°C
solubility 
≤20mg/ml in ethanol;25mg/ml in DMSO;25mg/ml in dimethyl formamide
form 
crystalline solid
color 
White to off-white
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GSK-2881078 Usage And Synthesis

Description

GSK2881078 is a selective androgen receptor modulator (SARM). It induces AR-mediated transcriptional activation in PC3(AR)2 cells (EC50 = 3.99 nM), an effect that can be inhibited by the non-steroidal AR antagonist bicalutamide .

Uses

GSK 2881078 is a selective androgen receptor modulator which can display agonistic properties in anabolic target tissues

References

[1]. https://newdrugapprovals.org/2016/06/14/gsk-2881078/

GSK-2881078Supplier

Yichang Chanod Biomedical Technology Co,LTD Gold
Tel
0717-6855399 15377615856
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sales@sndswyy.cn
HangZhou YuHao Chemical Technology Co., Ltd.
Tel
0571-82693216
Email
info@yuhaochemical.com
AdooQ Bioscience CHINA
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025-58849295 18951903616;
Email
info@adooq.cn
Shanghai Lollane Biological Technology Co.,Ltd.
Tel
021-52996696，15000506266 15000506266
PURE SYNMR INGREDIENTS LIMITED
Tel
021-26015538
Email
sven_shi@puresynmr.com
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GSK-2881078(1539314-06-1)Related Product Information