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Lanoconazole

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Lanoconazole Basic information

Product Name:
Lanoconazole
Synonyms:
  • LANOCONAZOLE
  • [4-(2-chloro-phenyl)-1,3-dithiolan-2-ylidene]-2-imidazol-1-yl-acetonitrile
  • (+-)-(e)-(4-(2-chlorophenyl)-1,3-dithiolan-2-ylidene)-1-imidazolylacetonitri
  • (e)-alpha-(4-(2-chlorophenyl)-1,3-dithiolan-2-ylidene)-1h-imidazole-1-aceton
  • 1h-imidazole-1-acetonitrile,alpha-(4-(2-chlorophenyl)-1,3-dithiolan-2-ylidene)
  • (E)-alpha-(4-(2-Chlorophenyl)-1,3-dithiolan-2-ylidene)-1H-imidazole-1-acetonitrile
  • 1H-Imidazole-1-acetonitrile, alpha-(4-(2-chlorophenyl)-1,3-dithiolan-2-ylidene)-, (E)-(+-)
  • (E)-2-[4-(2-Chlorophenyl)-1,3-dithiolane-2-ylidene]-2-(1-imidazolyl)acetonitrile
CAS:
101530-10-3
MF:
C14H10ClN3S2
MW:
319.83
EINECS:
635-180-5
Product Categories:
  • Intermediates & Fine Chemicals
  • Pharmaceuticals
Mol File:
101530-10-3.mol
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Lanoconazole Chemical Properties

Melting point:
141.50C
Boiling point:
477.6±55.0 °C(Predicted)
Density 
1.43±0.1 g/cm3(Predicted)
storage temp. 
2-8°C
solubility 
Chloroform (Slightly), Methanol (Slightly)
form 
Solid
pka
3.76±0.10(Predicted)
color 
White
CAS DataBase Reference
101530-10-3(CAS DataBase Reference)
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Safety Information

Hazard Codes 
Xn
Risk Statements 
22
WGK Germany 
3
RTECS 
NI3393500
Toxicity
LD50 in male, female mice, rats (mg/kg): 3224, 2715, 993, 652 orally; 2158, 1743, 1655, 2596 i.p.; >5000 both species s.c.; LD50 dermally in rats: >5000 mg/kg (Munt)
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Lanoconazole Usage And Synthesis

Description

Lanoconazole is a potent antifungal imidazole launched in Japan for the treatment of dermal mycoses. Lanoconazole is reported to be an inhibitor of ergosterol biosynthesis thus altering the ultra structure of the cell wall. It exhibits potent antifungal activity against a wide range of pathogenic fungi including yeast, dermatophytes, dermatiaceous fungi, dimorphic fungi, Aspergihs spp., Penici//ium spp., and Candida spp., being particularly active against Trichophyton spp.. It is considerably more potent than other agents of the same family such as bifonazole and clotrimazole. Clinical efficacy was demonstrated by remarkable improvements in skin symptoms of the patients with tinea pedis, tinea corporis and cruis, candidiasis or tinea versicolor.

Chemical Properties

Light-Yellow Crystals

Originator

Nihon Nohyaku (Japan)

Uses

Antifungal.

Definition

ChEBI: Lanoconazole is a conazole antifungal drug and an imidazole antifungal drug.

brand name

Astat

Lanoconazole Preparation Products And Raw materials

Raw materials

LanoconazoleSupplier

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