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Procaine penicilline G hydrate

Basic information Safety Supplier Related

Procaine penicilline G hydrate Basic information

Product Name:
Procaine penicilline G hydrate
Synonyms:
  • abbocillin-dc
  • crysticillin
  • despacilina
  • distaquaine
  • duracillin
  • enylacetamido)-,compd.with2-(diethylamino)ethylp-aminobenzoate(1:1),mono
  • flo-cillin
  • flo-cillinaqueous
CAS:
6130-64-9
MF:
C29H38N4O6S
MW:
570.71
EINECS:
612-112-2
Product Categories:
  • Agro-Products
  • Intermediates & Fine Chemicals
  • Pharmaceuticals
  • Sulfur & Selenium Compounds
Mol File:
6130-64-9.mol
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Procaine penicilline G hydrate Chemical Properties

Melting point:
106-110° (with decompn)
Density 
1.255-1.256
storage temp. 
Refrigerator
solubility 
Slightly soluble in water, sparingly soluble in ethanol (96 per cent).
form 
Solid
color 
White to Off-White
CAS DataBase Reference
6130-64-9(CAS DataBase Reference)
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Safety Information

Hazard Codes 
Xn
Risk Statements 
42/43
Safety Statements 
36
RTECS 
XH9450000
HS Code 
2941102000
Toxicity
LD50 s.c. in mice: 2.3 g/kg (Soehring)

MSDS

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Procaine penicilline G hydrate Usage And Synthesis

Description

Benzylpenicillin procaine was developed as a dilatorily acting benzylpenicillin, only slightly soluble in water. It has been used with peanut oil or carboxymethylcellulose as an oil suspension or an aqueous suspension, respectively .

Chemical Properties

White Solid

Uses

Procaine Penicillin G is a composed of the β-lactam antibiotic of Penicillin G and the sodium channel blocker Procaine. As an antibiotic, Penicillin G is noted to posses effectiveness mainly against gram-positive organisms. Procaine Penicillin G is used a growth stimulant for poultry.

Uses

Procaine penicilline G hydrate is a composed of the β-lactam antibiotic of Penicillin G and the sodium channel blocker Procaine. As an antibiotic, Penicillin G is noted to posses effectiveness mainly against gram-positive organisms. Procaine Penicillin G is used a growth stimulant for poultry.

brand name

Duracillin(Lilly); Pfizerpen (Pfizer).

Antimicrobial activity

The procaine salt of benzylpenicillin. Poorly soluble (1:200 in water). Administered intramuscularly as a suspension of crystals which slowly dissolve at the site of the injection.
It must not be given intravenously. Intramuscular administration produces a flat sustained plasma concentration of penicillin, which is much lower than that achieved by an equivalent dose of benzylpenicillin, with plasma levels still detectable 24 h later. An injection of 0.6 g yields a peak plasma concentration of 1–2 mg benzylpenicillin/L after 2–4 h. Free procaine is detectable in the plasma within 30 min.
Very severe and potentially fatal reactions resembling those of anaphylactic shock, but non-allergic in character, may occur, probably due to accidental entry into the vascular system at the site of injection and blockage of pulmonary and cerebral capillaries by crystals of the suspension. Reactions due to liberated procaine may include acute anxiety, hypertension, tachycardia, vomiting, audiovisual hallucinations and acute psychotic disturbance. The most severe reactions lead to convulsions and cardiac arrest. Other reactions are those to liberated benzylpenicillin.

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