2-(4-Iodophenyl)-6-methyl-1,3,6,2-dioxazaborocane-4,8-dione Chemical Properties

Melting point:

213-217 °C

Safety Information

Hazard Codes 

Xn

Risk Statements 

22

WGK Germany 

3

2-(4-Iodophenyl)-6-methyl-1,3,6,2-dioxazaborocane-4,8-dione Usage And Synthesis

Uses

4-Iodophenylboronic acid MIDA ester can be used:

• As a starting material to prepare rod-like hydrogen-bonded organic frameworks through Stille-coupling using 2,5-bis(trimethyltin)heterocycle, Pd(PPh₃)₄, and CuI.
• As a substrate in the C-H arylation reaction of pyroglutamic acid derivatives with aryl and heteroaryl iodides; catalyzed by the palladium catalyst.
• As a substrate in the synthesis of trifluoroborates, which are further converted to protected boronic acids.
• As a starting material in the synthesis of amino acid MIDA boronates as new building blocks by reacting with protected iodoalanine.

2-(4-Iodophenyl)-6-methyl-1,3,6,2-dioxazaborocane-4,8-dione(1257649-56-1)Related Product Information

• 4-Iodophenylboronic acid