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Indobufen

Basic information Safety Supplier Related

Indobufen Basic information

Product Name:
Indobufen
Synonyms:
  • 1-Oxo-2-[p-[(α-ethyl)carboxyMethyl]phenyl]isoindoline
  • 2-[p-(1-Oxo-2-isoindolinyl)phenyl]butyric Acid
  • K 2930
  • (+-)-butyricaci
  • 1-oxo-2-(p-((alpha-ethyl)carboxymethyl)phenyl)isoindoline
  • 4-(1,3-dihydro-1-oxo-2h-isoindol-2-yl)-alpha-ethyl-benzeneaceticacid
  • 2-[4-(1-OXO-1,3-DIHYDRO-ISOINDOL-2-YL)-PHENYL]-BUTYRIC ACID
  • lndobufen
CAS:
63610-08-2
MF:
C18H17NO3
MW:
295.34
EINECS:
264-364-4
Product Categories:
  • Amines
  • Aromatics
  • Heterocycles
  • Intermediates & Fine Chemicals
  • Pharmaceuticals
  • 63610-08-2
  • API
Mol File:
63610-08-2.mol
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Indobufen Chemical Properties

Melting point:
182-184°
Boiling point:
518.1±50.0 °C(Predicted)
Density 
1.275±0.06 g/cm3(Predicted)
storage temp. 
Keep in dark place,Sealed in dry,Room Temperature
solubility 
DMSO (Slightly), Methanol (Slightly)
form 
Solid
pka
4.39±0.10(Predicted)
color 
White
InChI
InChI=1S/C18H17NO3/c1-2-15(18(21)22)12-7-9-14(10-8-12)19-11-13-5-3-4-6-16(13)17(19)20/h3-10,15H,2,11H2,1H3,(H,21,22)
InChIKey
AYDXAULLCROVIT-UHFFFAOYSA-N
SMILES
O=C1C2C=CC=CC=2CN1C1C=CC(C(CC)C(=O)O)=CC=1
CAS DataBase Reference
63610-08-2(CAS DataBase Reference)
EPA Substance Registry System
Benzeneacetic acid, 4-(1,3-dihydro-1-oxo-2H-isoindol-2-yl)-.alpha.-ethyl- (63610-08-2)
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Indobufen Usage And Synthesis

Description

Indobufen is a platelet aggregation inhibitor related to the antiinflammatory agent indoprofen. It has shown clinical efficacy in peripheral artery disease, in prevention of deep vein thrombosis after myocardial infarction, and in blocking excercise-induced increase in platelet aggregation in angina patients.

Originator

Erbamont (Italy)

Uses

Indobufen is a platelet aggregation inhibitor. Indobufen is the anticoagulant drug and platelet aggregation inhibitor, which has anti-inflammatory analgesic effect. Indobufen is used as an antithrombotic.

Definition

ChEBI: Indobufen is a member of isoindoles.

brand name

IBUSTRIN

Clinical Use

A reversible but very potent inhibitor of platelet COX-1 activity, was shown to have comparable clinical efficacy to that of aspirin in prevention of DVT after myocardial infarction and in blocking exercise-induced increase in platelet aggregation. In the secondary prevention of thromboembolic events, 100 or 200 mg of indobufen twice daily is as effective as warfarin or aspirin in patients with or without atrial fibrillation. Currently, indobufen is only available for routine clinical use in Europe.

Indobufen Preparation Products And Raw materials

Raw materials

IndobufenSupplier

Hubei Chenxin Pharmaceutical Co., Ltd. Gold
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Huadong Medicine (Xi'an)Bodyguard Pharmaceutical Co.,Ltd. Gold
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029-86638659 18109298458
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Hubei Weideli Chemical Reagent Co.,Ltd. Gold
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027-59222918 13385289472
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J & K SCIENTIFIC LTD.
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010-82848833 400-666-7788
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jkinfo@jkchemical.com
Wuhan Jiakai Long Technology Development Co., Ltd.
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027-88422011