Basic information Safety Supplier Related

N4-Benzoyl-5'-O-DMT-2'-O-methyl-5-methylcytidine 3'-CE phosphoramidite

Basic information Safety Supplier Related

N4-Benzoyl-5'-O-DMT-2'-O-methyl-5-methylcytidine 3'-CE phosphoramidite Basic information

Product Name:
N4-Benzoyl-5'-O-DMT-2'-O-methyl-5-methylcytidine 3'-CE phosphoramidite
Synonyms:
  • N4-Benzoyl-5'-O-DMT-2'-O-methyl-5-methylcytidine 3'-CE phosphoramidite
  • N4-Acetyl-5-methyl-5'-O-(4,4'-dimethoxytrityl)-2'-O-methyl-5-Methylcytidine-3'- CE-cyanoethyl Phosphoramidite
  • N-Benzoyl-5'-O-[bis(4-methoxyphenyl)phenylmethyl]-2'-O-(2-methoxyethyl)cytidine 3'-[2-cyanoethyl bis(1-methylethyl)phosphoramidite]
  • 2'-O-MOE-C(Bz)-CE Phosphoramidite
  • 2'-O-MOE-C(Bz)-3'-phosphoramidite
  • 2'-O-MOE-Bz-C Phosphoramidite
  • Cytidine, N-benzoyl-5'-O-[bis(4-methoxyphenyl)phenylmethyl]-2'-O-(2-methoxyethyl)-, 3'-[2-cyanoethyl bis(1-methylethyl)phosphoramidite] (9CI)
  • N4-Bz-5’-O-DMTr-2’-O-(2-methoxyethyl)cytidine-3’-CED-phosphoramidite
CAS:
251647-54-8
MF:
C49H58N5O10P
MW:
908
Mol File:
251647-54-8.mol
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N4-Benzoyl-5'-O-DMT-2'-O-methyl-5-methylcytidine 3'-CE phosphoramidite Chemical Properties

storage temp. 
Store at -20°C
form 
Solid
pka
8.57±0.20(Predicted)
color 
White to light yellow
InChIKey
IAFVTVZPQIFRAU-STEDOTHVNA-N
SMILES
C(C1C=CC=CC=1)(C1C=CC(OC)=CC=1)(C1C=CC(OC)=CC=1)OC[C@H]1O[C@@H](N2C=CC(NC(C3C=CC=CC=3)=O)=NC2=O)[C@H](OCCOC)[C@@H]1OP(OCCC#N)N(C(C)C)C(C)C |&1:25,27,44,50,r|
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N4-Benzoyl-5'-O-DMT-2'-O-methyl-5-methylcytidine 3'-CE phosphoramidite Usage And Synthesis

Uses

2'-O-MOE-rC is a 2'-O-MOE modified nucleoside. 2'-O-MOE-rC can be used for synthesis of DNA[1][2].

References

[1] Prakash TP, et al. Comparing in vitro and in vivo activity of 2'-O-[2-(methylamino)-2-oxoethyl]- and 2'-O-methoxyethyl-modified antisense oligonucleotides. J Med Chem. 2008 May 8;51(9):2766-76. DOI:10.1021/jm701537z
[2] Li M, et al. Synthesis and cellular activity of stereochemically-pure 2'-O-(2-methoxyethyl)-phosphorothioate oligonucleotides. Chem Commun (Camb). 2017 Jan 3;53(3):541-544. DOI:10.1039/c6cc08473g

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