Basic information Safety Supplier Related
ChemicalBook >  Product Catalog >  API >  Antipyretic analgesics >  Ubrogepant

Ubrogepant

Basic information Safety Supplier Related

Ubrogepant Basic information

Product Name:
Ubrogepant
Synonyms:
  • Ubrogepant
  • MK-1602
  • MK-1602 Ubrogepant
  • Spiro[6H-cyclopenta[b]pyridine-6,3'-[3H]pyrrolo[2,3-b]pyridine]-3-carboxamide, 1',2',5,7-tetrahydro-N-[(3S,5S,6R)-6-methyl-2-oxo-5-phenyl-1-(2,2,2-trifluoroethyl)-3-piperidinyl]-2'-oxo-, (3'S)-
  • Ubrogepant API
  • Ubrogepant D5
  • (S)-N-((3S,5S,6R)-6-methyl-2-oxo-5-phenyl-1-(2,2,2-trifluoroethyl)piperidin-3-yl)-2'-oxo-1',2',5,7-tetrahydrospiro[cyclopenta[b]pyridine-6,3'-pyrrolo[2,3-b]pyridine]-3-carboxamide
  • MK1602,MK 1602,Ubrogepant,inhibit,Inhibitor,Calcitonin gene-related peptide receptor,CGRP Receptor
CAS:
1374248-77-7
MF:
C29H26F3N5O3
MW:
549.54
Product Categories:
  • API
  • 1374248-77-7
Mol File:
1374248-77-7.mol
More
Less

Ubrogepant Chemical Properties

Boiling point:
729.4±60.0 °C(Predicted)
Density 
1.45±0.1 g/cm3(Predicted)
storage temp. 
Store at -20°C
solubility 
Soluble in DMSO
form 
Solid
pka
11.08±0.20(Predicted)
color 
White to off-white
InChIKey
DDOOFTLHJSMHLN-ZQHRPCGSSA-N
SMILES
C12C[C@@]3(C(=O)NC4=NC=CC=C43)CC1=CC(C(N[C@H]1C[C@@H](C3=CC=CC=C3)[C@@H](C)N(CC(F)(F)F)C1=O)=O)=CN=2
More
Less

Ubrogepant Usage And Synthesis

Uses

Ubrogepant, is a new drug possible used for the treatment of migraine.

Synthesis

Synthesis route of Ubrogepant

in vivo

Ubrogepant (0.06-100 μg/kg; intravenous injection; 1-3 times) inhibits Capsaicin (HY-10448)-induced dermal vasodilation in a concentration- and time-dependent manner in rhesus monkeys with an EC50 of 3.19 nM[1].

UbrogepantSupplier

Jiangsu Vcare PharmaTech Co., Ltd. Gold
Tel
025-58741518 13327700685
Email
sales@vcarepharmatech.com
Kaifeng Mingren Pharmaceutical Co.,LTD Gold
Tel
0371-65741762
Email
sales@hasunny.com
ChengDu TongChuangYuan Pharmaceutical Co.Ltd Gold
Tel
028-83379370 13880556291
Email
tcy@tcypharm.com
J & K SCIENTIFIC LTD.
Tel
18210857532; 18210857532
Email
jkinfo@jkchemical.com
Anhui Lianchuang Biological Medicine Co.,Ltd
Tel
0551-68779238 18056025720
Email
sales3@lcywhx.com