3-Aminocarbonylphenylboronic acid Chemical Properties

Melting point:

221-226 °C

Boiling point:

408.1±47.0 °C(Predicted)

Density 

1.32±0.1 g/cm3(Predicted)

storage temp. 

2-8°C

solubility 

soluble in Methanol

pka

7.84±0.10(Predicted)

form 

Solid

color 

White to off-white

CAS DataBase Reference

351422-73-6(CAS DataBase Reference)

Safety Information

Hazard Codes 

Xi,Xn

Risk Statements 

22-36/37/38-20/21/22

Safety Statements 

26-36-24/25

WGK Germany 

3

Hazard Note 

Corrosive

HazardClass 

IRRITANT

HS Code 

29310095

3-Aminocarbonylphenylboronic acid Usage And Synthesis

Chemical Properties

White to brown solid

Uses

Reactant involved in the synthesis of a variety of inhibitors including:

• Orally active phosphodiesterase 10A inhibitors
• Pyrimidine derivatives as TpI2 kinase inhibitors
• Peptidomimetic inhibitors of STAT3 protein

• Oxidative cross-coupling with mercaptoacetylenes
• Trifluoromethylation via a Collidine trifluoromethylating agent
• Suzuki cross-coupling reactions

Uses

Reactant involved in the synthesis of a variety of inhibitors including:• ;Orally active phosphodiesterase 10A inhibitors1• ;Pyrimidine derivatives as TpI2 kinase inhibitors2• ;Peptidomimetic inhibitors of STAT3 protein3Reactant involved in:• ;Oxidative cross-coupling with mercaptoacetylenes4• ;Trifluoromethylation via a Collidine trifluoromethylating agent5• ;Suzuki cross-coupling reactions6

Uses

suzuki reaction

3-Aminocarbonylphenylboronic acid(351422-73-6)Related Product Information

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• P-AMINOBENZAMIDE GLUTAMIC ACID
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• 3-(4-FLUOROPHENYL)AMINOCARBONYLPHENYLBORONIC ACID PINACOL ESTER
• 2-AMINOCARBONYLPHENYLBORONIC ACID
• 4-(PYRIDIN-2-YL)AMINOCARBONYLPHENYLBORONIC ACID
• 4-AMINOCARBONYLPHENYLBORONIC ACID, PINACOL ESTER