Basic information Safety Supplier Related
ChemicalBook >  Product Catalog >  Analytical Chemistry >  Standard >  Pharmaceutical Impurity Reference Standards >  Dolutegravir 2-Desfluoro Impurity

Dolutegravir 2-Desfluoro Impurity

Basic information Safety Supplier Related

Dolutegravir 2-Desfluoro Impurity Basic information

Product Name:
Dolutegravir 2-Desfluoro Impurity
Synonyms:
  • 2H-Pyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazine-9-carboxamide, N-[(4-fluorophenyl)methyl]-3,4,6,8,12,12a-hexahydro-7-hydroxy-4-methyl-6,8-dioxo-, (4R,12aS)-/Dolutegravir impurity
  • Dolutegravir impurity 4/Defluoro Dolutegravir/(4R,12aS)-N-(4-Fluorobenzyl)-7-hydroxy-4-methyl-6,8-dioxo-3,4,6,8,12,12a-hexahydro-2H-pyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazine-9-carboxamide
  • Dolutegravir Impurity G
  • Dolutegravir 2-Desfluoro Impurity
  • 2H-Pyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazine-9-carboxamide, N-[(4-fluorophenyl)methyl]-3,4,6,8,12,12a-hexahydro-7-hydroxy-4-methyl-6,8-dioxo-, (4R,12aS)-
  • (4R,12aS)-N-(4-fluorobenzyl)-7-hydroxy-4-methyl-6,8-dioxo-3,4,6,8,12,12a-hexahydro-2H-pyrido[1',2':4,5]pyrazino[2,1-b][1,3]oxazine-9-carboxamide
  • Dolutegravir Impurity 47
  • Dolutegravir Impurity 50
CAS:
1863916-88-4
MF:
C20H20FN3O5
MW:
401.39
Mol File:
1863916-88-4.mol
More
Less

Dolutegravir 2-Desfluoro Impurity Chemical Properties

Boiling point:
675.7±55.0 °C(Predicted)
Density 
1.49±0.1 g/cm3(Predicted)
solubility 
DMSO (Slightly), Methanol (Slightly, Heated)
form 
Solid
pka
4.50±1.00(Predicted)
color 
Off-White to Light Brown
More
Less

Dolutegravir 2-Desfluoro Impurity Usage And Synthesis

Uses

Defluoro Dolutegravir is an impurity of Dolutegravir (D528800), a second generation HIV-1 integrase strand transfer inhibitor. Dolutegravir is currently in Phase III clinical trials for the treatment of HIV infection. Dolutegravir has been shown to potently inhibit HIV replication in cells such as peripheral blood mononuclear cells (PBMCs), MT-4 cells and CIP4 cells infected with a self-inactivating PHIV lentiviral vector.

Dolutegravir 2-Desfluoro ImpuritySupplier

Shenzhen Roark Pharma-Tec Co., Ltd. Gold
Tel
13128912434
Email
2880126944@qq.com
Beijing Comparison Pharmaceutical Technology Co., Ltd
Tel
010-010-52878169 15801002657
Email
sales@bjcomparison.com
ChemStrong Scientific Co.,Ltd
Tel
0755-0755-66853366 13670046396
Email
sales@chem-strong.com
Shanghai CR Corporation Limited
Tel
021-80270511; 4006653949
Email
fred.wen@crcorporation.cn
CR Corporation Limited
Tel
+8613062833949
Email
fred.wen@crcorporation.cn