Basic information Safety Supplier Related

ALLOPURINOL RIBOSIDE

Basic information Safety Supplier Related

ALLOPURINOL RIBOSIDE Basic information

Product Name:
ALLOPURINOL RIBOSIDE
Synonyms:
  • 1-BETA-D-RIBOFURANOSYL-1H-PYRAZOLO[3,4-D]PYRIMIDINE-4-ONE
  • 1-BETA-D-RIBOFURANOSYLPYRAZOLO[3,4-D]PYRIMIDIN-4-ONE
  • ALLOPURINOL RIBOSIDE
  • 8-AZA-7-DEAZAINOSINE
  • 1-β-d-ribofuranosyl-1h-pyrazolo[3,4-d]pyrimidine-4-one
  • 1-[(2S,3S,4R,5R)-3,4,5,6-tetrahydroxyoxan-2-yl]-2H-pyrazolo[4,5-e]pyrimidin-4-one
  • 1,5-Dihydro-1-β-D-ribofuranosyl-4H-pyrazolo[3,4-d]pyrimidin-4-one
  • Allopurinol ribonucleoside
CAS:
16220-07-8
MF:
C10H12N4O5
MW:
268.23
Mol File:
16220-07-8.mol
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ALLOPURINOL RIBOSIDE Chemical Properties

Boiling point:
715.0±60.0 °C(Predicted)
Density 
2.08±0.1 g/cm3(Predicted)
storage temp. 
2-8°C
solubility 
DMSO:5.0(Max Conc. mg/mL);18.64(Max Conc. mM)
PBS (pH 7.2):5.0(Max Conc. mg/mL);18.64(Max Conc. mM)
form 
A solid
pka
8.65±0.10(Predicted)
color 
White to off-white
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Safety Information

WGK Germany 
3

MSDS

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ALLOPURINOL RIBOSIDE Usage And Synthesis

Uses

Allopurinol riboside is a structural isomer of hypoxanthine.

Definition

ChEBI: A nucleoside analogue that is allopurinol with a beta-D-ribofuranosyl moiety at the 1-position.

in vivo

Allopurinol riboside peaks in plasma 1.6 hours after administration, has an elimination half-life of 3 hours, and steady-state concentrations in the therapeutic range[3]. After oral administration, unexpectedly low levels of allopurinol riboside in plasma are attributable to incomplete absorption and rapid renal clearance. Probenecid reduces the renal clearance of allopurinol riboside, extends the half-life of allopurinol riboside in plasma, and triples the levels of allopurinol riboside in plasma[4].

IC 50

Leishmania

ALLOPURINOL RIBOSIDESupplier

Beijing Jin Ming Biotechnology Co., Ltd.
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010-60605840 18892239720
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psaitong@jm-bio.com
Shenzhen Regent Biochemical Technology Co., Ltd.
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0755-85201366 18938635012
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sales@regentsciences.com
Aikon International Limited
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025-58859352 18068836627
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dt3@aikonchem.com
Jinan Yaoyan Pharmaceutical Co., Ltd.
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Shenzhen Botel Biotechnology Co. Ltd.
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13316949107 13316968096
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