Basic information Safety Supplier Related
ChemicalBook >  Product Catalog >  Analytical Chemistry >  Standard >  Pharmaceutical Impurity Reference Standards >  Crisaborole intermediate

Crisaborole intermediate

Basic information Safety Supplier Related

Crisaborole intermediate Basic information

Product Name:
Crisaborole intermediate
Synonyms:
  • 5-(4-(hydroxymethyl)phenoxy)benzo[c][1,2]oxaborol-1(3H)-ol
  • Crisaborole Impurity 59
  • 5-(4-(Hydroxylmethyl)phenoxy)benzo[c][1,2]oxaborol-1-(3H)-ol
  • Crisaborole Impurity 37
  • Crisaborole Impurity 28
  • Benzenemethanol, 4-[(1,3-dihydro-1-hydroxy-2,1-benzoxaborol-5-yl)oxy]-
  • Creborol Impurity 28
CAS:
1187188-60-8
MF:
C14H13BO4
MW:
256.06
Mol File:
1187188-60-8.mol
More
Less

Crisaborole intermediate Chemical Properties

Boiling point:
432.1±55.0 °C(Predicted)
Density 
1.33±0.1 g/cm3(Predicted)
pka
7.05±0.20(Predicted)
More
Less

Crisaborole intermediate Usage And Synthesis

Uses

5-(4-(Hydroxyl Methyl)phenoxy)benzo[c][1,2]oxaborol-1-(3H)-ol is an impurity for Crisaborole(H947928). Crisaborole is a series of phenoxy benzoxaboroles were synthesized and screened for their inhibitory activity against PDE4 and cytokine release. 5-?(4-?Cyanophenoxy)?-?2,?3-?dihydro-?1-?hydroxy-?2,?1-?benzoxaborole (AN2728) showed potent activity both in vitro and in vivo. AN2728 is being studied as an anti-inflammatory agent.

Crisaborole intermediateSupplier

Beijing Comparison Pharmaceutical Technology Co., Ltd
Tel
010-010-52878169 15801002657
Email
sales@bjcomparison.com
ChemStrong Scientific Co.,Ltd
Tel
0755-0755-66853366 13670046396
Email
sales@chem-strong.com
Hubei Yangxin Medical Technology Co., Ltd.
Tel
15374522761
Email
3003392093@qq.com
TOSUN PHARM
Tel
020-61855200 13326451905
Email
260366801@qq.com
ANHUI WITOP BIOTECH CO., LTD
Tel
+8615255079626
Email
eric@witopchemical.com