ChemicalBook > Product Catalog > API > Synthetic Anti-infective Drugs > Antifungal Drugs > SAPERCONAZOLE
SAPERCONAZOLE
SAPERCONAZOLE Basic information
- Product Name:
- SAPERCONAZOLE
- Synonyms:
-
- SAPERCONAZOLE
- R-66905
- (+-)-1-sec-Butyl-4-(p-(4-(p-(((2R*,4S*)-2-(2,4-difluorophenyl)-2-(1H-1 ,2,4-triazol-1-ylmethyl)-1,3-dioxolan-4-yl)methoxy)phenyl)-1-piperazin yl)phenyl)-delta(sup 2)-1,2,4-triazolin-5-one
- 4-[4-[4-[4-[[2-(2，4-Difluorophenyl)-2-(1H-1，2，4-triazol-1-yl-methyl)-1，3-dioxolan-4-y1]methoxyl]phenyl]-1-piperazinyl]phenyl]-2，4-dihydrcr2-(1-methylpropyl)-3H-1，2，4-triazol-3-one
- 2-(1H-1,2,4-Triazol-1-ylmethyl)-2-(2,4-difluorophenyl)-4-[[4-[4-[4-[[2-(1-methylpropyl)-2,3-dihydro-3-oxo-4H-1,2,4-triazol]-4-yl]phenyl]piperazin-1-yl]phenoxy]methyl]-1,3-dioxolane
- 2-sec-Butyl-4-[4-[4-[4-[[2-(1H-1,2,4-triazole-1-ylmethyl)-2-(2,4-difluorophenyl)-1,3-dioxolane-4-yl]methoxy]phenyl]-1-piperazinyl]phenyl]-2,4-dihydro-3H-1,2,4-triazole-3-one
- a-(2 4-DIFLUOROPHENYL)-a-(1H-1 2 4-TRAIZ OL-1-YLMETHYL)-1H-1 2 4-TRIAZOLE-1-ETHAN OL(FLUCONAZOLE)
- 3H-1,2,4-Triazol-3-one, 4-[4-[4-[4-[[2-(2,4-difluorophenyl)-2-(1H-1,2,4-triazol-1-ylmethyl)-1,3-dioxolan-4-yl]methoxy]phenyl]-1-piperazinyl]phenyl]-2,4-dihydro-2-(1-methylpropyl)-
- CAS:
- 110588-57-3
- MF:
- C35H38F2N8O4
- MW:
- 672.72
- Mol File:
- 110588-57-3.mol
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SAPERCONAZOLE Chemical Properties
- Melting point:
- 189.5°
- Boiling point:
- 812.5±75.0 °C(Predicted)
- Density
- 1.37±0.1 g/cm3(Predicted)
- storage temp.
- 2-8°C
- solubility
- Soluble in DMSO
- form
- Solid
- pka
- 6.47±0.40(Predicted)
- color
- Off-white to light yellow
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SAPERCONAZOLE Usage And Synthesis
Uses
Antifungal.
Uses
Saperconazole is an analog of Itraconazole (I937500), an orally active antimycotic structurally related to Ketoconazole.
in vivo
All control pigeons infect with A. fumigatus die within 2 to 5 days. They have necrotic foci in the lungs, air sacs, liver, spleen, and kidneys. These organs are highly positive by histology and oncultures. Saperconazole administered at 2.5 mg/kg is not active, but when it is given at 5 or 10 mg/kg, 92 or 100%, respectively, survive and organ cultures are negative. No drug-related side effects are observed in the pigeons[2].
SAPERCONAZOLE Preparation Products And Raw materials
Raw materials
SAPERCONAZOLESupplier
LGM Pharma
- Tel
- 1-(800)-881-8210
- inquiries@lgmpharma.com
Clearsynth Labs Limited
- Tel
- +91-22-26355700
- info@clearsynth.com
Fan De(Beijing) Biotechnology Co., Ltd.
- Tel
- 15911056312
- liming@bio-fount.com
Hangzhou Synstar pharmaceutical Technology CO.,Ltd
- Tel
- 0571-85361029
- synstar518@163.com
TargetMol Chemicals Inc.
- Tel
- +1-781-999-5354 +1-00000000000
- marketing@targetmol.com
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SAPERCONAZOLE(110588-57-3)Related Product Information
- 2-AMINO-1-(2-FLUORO-PHENYL)-ETHANOL
- 2,4-dihydro-4-[4-[4-(4-methoxyphenyl)piperazin-1-yl]phenyl]-3H-1,2,4-triazol-3-one
- 1-(4-AMINOPHENYL)-4-(4-METHOXYPHENYL)PIPERAZINE
- 1-(4-Aminophenyl)-4-(4-hydroxyphenyl)piperazine
- 2,4-Dihydro-4-[4-[4-(4-methoxyphenyl)-1-piperazinyl]phenyl]-2-(1-methylpropyl)-3H-1,2,4-triazol-3-one
- 1-(4-ETHOXYPHENYL)PIPERAZINE
- 2,4-DIHYDRO-4-[(4-(4-HYDROXYPHENYL)-1-PIPERAZINYL)PHENYL]-2-(1-METHYLPROPYL)-3H-1,2,4-TRIAZOLE-3-ONE
- SAPERCONAZOLE
- Posaconazole
- (R)-1-(2-FLUOROPHENYL)ETHANOL
- 1,4-DIPHENYLPIPERAZINE
- 2,4-Dihydro-4-phenyl-3H-1,2,4-triazol-3-one
- 1,2-Propanediol, 3-(p-(dimethylamino)phenoxy)-
- Benzeneethanamine, 2,4-difluoro- (9CI)
- Dimethyl-(4-piperazin-1-yl-phenyl)-amine
- 2-amino-1-(2,4-difluorophenyl)ethanol
- (S)-1-(2-FLUOROPHENYL)ETHANOL
- 1-[4-(2-METHOXY-ETHOXY)-PHENYL]-PIPERAZINE