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Pyrazolo[1,5-a]pyridine-3-carbonitrile, 4-(6-fluoro-3-pyridinyl)-6-hydroxy-

Basic information Safety Supplier Related

Pyrazolo[1,5-a]pyridine-3-carbonitrile, 4-(6-fluoro-3-pyridinyl)-6-hydroxy- Basic information

Product Name:
Pyrazolo[1,5-a]pyridine-3-carbonitrile, 4-(6-fluoro-3-pyridinyl)-6-hydroxy-
Synonyms:
  • Pyrazolo[1,5-a]pyridine-3-carbonitrile, 4-(6-fluoro-3-pyridinyl)-6-hydroxy-
  • 4-(6-Fluoropyridin-3-yl)-6-hydroxypyrazolo[1,5-a]pyridine-3-carbonitrile
  • 4-(6-fluoro-3-pyridyl)-6-hydroxy-pyrazolo[1,5-a]pyridine-3-carbonitrile
  • 4-(6- Fluoropyridin -3-y1)-6- hydroxypyrazolo [1,5- a ] pyridine -3- carbonitrile
  • 4-(6-Fluoro-3-pyridinyl)-6-hydroxypyrazolo[1,5-a]pyridine-3-carbonitrile
CAS:
2222654-09-1
MF:
C13H7FN4O
MW:
254.22
Mol File:
2222654-09-1.mol
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Pyrazolo[1,5-a]pyridine-3-carbonitrile, 4-(6-fluoro-3-pyridinyl)-6-hydroxy- Chemical Properties

InChI
InChI=1S/C13H7FN4O/c14-12-2-1-8(5-16-12)11-3-10(19)7-18-13(11)9(4-15)6-17-18/h1-3,5-7,19H
InChIKey
VOTPTQNCWJNQGK-UHFFFAOYSA-N
SMILES
C12=C(C#N)C=NN1C=C(O)C=C2C1=CC=C(F)N=C1
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Pyrazolo[1,5-a]pyridine-3-carbonitrile, 4-(6-fluoro-3-pyridinyl)-6-hydroxy- Usage And Synthesis

Uses

Pyrazolo[1,5-a]pyridine-3-carbonitrile, 4-(6-fluoro-3-pyridinyl)-6-hydroxy- is a pharmaceutical intermediate that can be used to prepare serpatinib.

Synthesis

Pyrazolo[1,5-a]pyridine-3-carbonitrile, 4-(6-fluoro-3-pyridinyl)-6-hydroxy- can be prepared from (E)-4-bromo-6-methoxypyrazolo[1,5-a]pyridine-3-carboxaldehyde oxime by a five-step reaction.

Pyrazolo[1,5-a]pyridine-3-carbonitrile, 4-(6-fluoro-3-pyridinyl)-6-hydroxy-Supplier

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