Basic information Brand Name(s) in US Safety Supplier Related
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Difluoxacin hydrochloride

Basic information Brand Name(s) in US Safety Supplier Related

Difluoxacin hydrochloride Basic information

Product Name:
Difluoxacin hydrochloride
Synonyms:
  • VETRANAL
  • 6-FLUORO-1-(4-FLUOROPHENYL)-1,4-DIHYDRO-7-(4-METHYLPIPERAZINO)-4-OXO-3-QUINOLINECARBOXYLIC ACID HYDROCHLORIDE
  • DIFLUOXACIN HYDROCHLORIDE
  • DIFLOXACIN HCL
  • DIFLOXACIN HYDROCHLORIDE
  • Difluoxacin HCL
  • 6-Fluoro-1-(4-fluorophenyl)-7-(4-methylpiperazin-1-yl)-4-oxoquinoline-3-carboxylic acid hydrochloride
  • 3-Quinolinecarboxylic acid, 6-fluoro-1-(4-fluorophenyl)-1,4-dihydro-7-(4-methyl-1-piperazinyl)-4-oxo-, monohydrochloride
CAS:
91296-86-5
MF:
C21H20ClF2N3O3
MW:
435.85
EINECS:
1806241-263-5
Product Categories:
  • DICURAL
  • Active Pharmaceutical Ingredients
  • Chiral Reagents
  • Inhibitors
  • Intermediates & Fine Chemicals
  • Pharmaceuticals
  • API
Mol File:
91296-86-5.mol
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Difluoxacin hydrochloride Chemical Properties

Melting point:
>245°C (dec.)
storage temp. 
Inert atmosphere,Room Temperature
solubility 
Soluble in aqueous buffer
form 
powder
color 
White to off-white
InChI
InChI=1S/C21H19F2N3O3.ClH/c1-24-6-8-25(9-7-24)19-11-18-15(10-17(19)23)20(27)16(21(28)29)12-26(18)14-4-2-13(22)3-5-14;/h2-5,10-12H,6-9H2,1H3,(H,28,29);1H
InChIKey
JFMGBGLSDVIOHL-UHFFFAOYSA-N
SMILES
C12C=C(C(F)=CC=1C(C(C(=O)O)=CN2C1=CC=C(F)C=C1)=O)N1CCN(C)CC1.Cl
CAS DataBase Reference
91296-86-5(CAS DataBase Reference)
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Safety Information

WGK Germany 
3
RTECS 
VB2008975
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Difluoxacin hydrochloride Usage And Synthesis

Brand Name(s) in US

Dicural

Description

Difloxacin is a fluoroquinolone antibiotic. It is active against isolates of anaerobic bacteria, including B. fragilis, as well as Fusobacterium and Actinomyces species with MIC values ranging from ≤0.125 to 8 μg/ml. It eliminates E. coli and B. fragilis infection in a rat intra-abdominal abscess model when administered at a dose of 40 mg/kg three times per day.

Chemical Properties

Off-White to Pale Yellow Solid

Uses

antibacterial, DNA gyrase inhibitor

Uses

A quinolone antibacterial compound. Structurally related to norfloxacin

Uses

A fluoroquinolone antibacterial structurally related to norfloxacin.

References

[1] M B BANSAL  H T. Activity of difloxacin (A-56619) and A-56620 against clinical anaerobic bacteria in vitro.[J]. Antimicrobial Agents and Chemotherapy, 1987, 31 4: 619-621. DOI: 10.1128/aac.31.4.619
[2] H THADEPALLI  S K C  S V Gollapudi. Therapeutic evaluation of difloxacin (A-56619) and A-56620 for experimentally induced Bacteroides fragilis-associated intra-abdominal abscess.[J]. Antimicrobial Agents and Chemotherapy, 1986, 30 4: 574-576. DOI: 10.1128/aac.30.4.574

Difluoxacin hydrochlorideSupplier

Xiamen Weijia Pharma Co., Ltd Gold
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