Basic information Safety Supplier Related
ChemicalBook >  Product Catalog >  Organic Chemistry >  Organosulfur compounds >  4-(2-(4,4-Dimethyl-4,5-dihydrooxazol-2-yl)propan-2-yl)phenethyl 4-methylbenzenesulfonate

4-(2-(4,4-Dimethyl-4,5-dihydrooxazol-2-yl)propan-2-yl)phenethyl 4-methylbenzenesulfonate

Basic information Safety Supplier Related

4-(2-(4,4-Dimethyl-4,5-dihydrooxazol-2-yl)propan-2-yl)phenethyl 4-methylbenzenesulfonate Basic information

Product Name:
4-(2-(4,4-Dimethyl-4,5-dihydrooxazol-2-yl)propan-2-yl)phenethyl 4-methylbenzenesulfonate
Synonyms:
  • Benzeneethanol, 4-[1-(4,5-dihydro-4,4-dimethyl-2-oxazolyl)-1-methylethyl]-, 4-methylbenzenesulfonate (ester)
  • 4-(2-(4,4-Dimethyl-4,5-dihydrooxazol-2-yl)propan-2-yl)phenethyl 4-methylbenzenesulfonate
  • 2-[4-[1-(4,4-dimethyl-5H-oxazol-2-yl)-1-methyl-ethyl]phenyl]ethyl 4-methylbenzenesulfonate
  • Bilastine impurity C
  • 2-[4-[1-(4,4-Dimethyl-5H-Oxazol-2-Yl)-1- Methyl-Ethyl]Phenyl
  • Benzeneethanol, 4-[1-(4,5-dihydro-4,4-dimethyl-2-oxazolyl)-1-methylethyl]-, 1-(4-methylbenzenesulfonate)
  • 4 - (2 - (4,4-dimethyl-4,5-dihydroxazol-2-yl) propyl-2-yl) phenylethyl 4-methylbenzene sulfonate
  • 4-(2-((4,4-dimethyl-4,5-dihydroxyoxazol-2-yl)propan-2yl)phenethyl-4-methylbenzenesulfonate
CAS:
202189-76-2
MF:
C23H29NO4S
MW:
415.55
EINECS:
606-467-2
Mol File:
202189-76-2.mol
More
Less

4-(2-(4,4-Dimethyl-4,5-dihydrooxazol-2-yl)propan-2-yl)phenethyl 4-methylbenzenesulfonate Chemical Properties

Boiling point:
545.1±45.0 °C(Predicted)
Density 
1.14±0.1 g/cm3(Predicted)
vapor pressure 
0Pa at 25℃
storage temp. 
2-8°C
solubility 
soluble in Dichloromethane;
pka
5.78±0.70(Predicted)
Water Solubility 
5.717μg/L at 25℃
InChI
InChI=1S/C23H29NO4S/c1-17-6-12-20(13-7-17)29(25,26)28-15-14-18-8-10-19(11-9-18)23(4,5)21-24-22(2,3)16-27-21/h6-13H,14-16H2,1-5H3
InChIKey
BGUOPDZOVDIWLE-UHFFFAOYSA-N
SMILES
C(C1C=CC(CCOS(C2C=CC(C)=CC=2)(=O)=O)=CC=1)(C1OCC(C)(C)N=1)(C)C
LogP
6.6
More
Less

4-(2-(4,4-Dimethyl-4,5-dihydrooxazol-2-yl)propan-2-yl)phenethyl 4-methylbenzenesulfonate Usage And Synthesis

Uses

4-(2-(4,4-Dimethyl-4,5-dihydrooxazol-2-yl)propan-2-yl)phenethyl 4-methylbenzenesulfonate (or Benzeneethanol, 4-[1-(4,5-dihydro-4,4-dimethyl-2-oxazolyl)-1-methylethyl]-, 4-methylbenzenesulfonate (ester)) is an intermediate used in the synthesis of Bilastine-d6 (B385002), which is labelled Bilastine. It is a novel, nonsedating H1-antihistamine developed for symptomatic treatment of allergic rhinitis and chronic idiopathic urticaria.

4-(2-(4,4-Dimethyl-4,5-dihydrooxazol-2-yl)propan-2-yl)phenethyl 4-methylbenzenesulfonateSupplier

Anhui Dexinjia Biopharm Co., Ltd Gold
Tel
0531-82375878 15269101859
Email
2710825968@qq.com
Shanghai Joiny Pharmaceutical Co.,Ltd. Gold
Tel
13681955282
Email
gyd@joiny-pharma.com
Adamas Reagent, Ltd.
Tel
400-6009262 16621234537
Email
chenyj@titansci.com
Shanghai Boc Chemical Co.,Ltd
Tel
021-34975603-808 18721111801
Email
sales@bocpharma.com
Changzhou Wanyao Biotechnology Co., Ltd.
Tel
0519-89185693 15312551983
Email
2410037592@qq.com