Basic information Safety Supplier Related
ChemicalBook >  Product Catalog >  Pharmaceutical intermediates >  Heterocyclic compound >  Piperazine compounds >  Dropropizine

Dropropizine

Basic information Safety Supplier Related

Dropropizine Basic information

Product Name:
Dropropizine
Synonyms:
  • 3-(4-phenyl-1-piperazinyl)-2-propanediol
  • catabex
  • dipropizine
  • ditustat
  • dopropizin
  • katril
  • larylin
  • 1,2-PROPANEDIOL, 3-(4-PHENYL-1-PIPERAZINYL)-
CAS:
17692-31-8
MF:
C13H20N2O2
MW:
236.31
EINECS:
241-683-7
Product Categories:
  • Aromatics
  • Heterocycles
  • Intermediates & Fine Chemicals
  • Pharmaceuticals
Mol File:
17692-31-8.mol
More
Less

Dropropizine Chemical Properties

Melting point:
105° (Morren); mp 108° (Bourdais)
Boiling point:
205 °C(Press: 1 Torr)
Density 
1.168±0.06 g/cm3(Predicted)
storage temp. 
Sealed in dry,Room Temperature
solubility 
Chloroform (Sparingly), Methanol (Slightly)
form 
Solid
pka
14.21±0.20(Predicted)
color 
White to Off-White
CAS DataBase Reference
17692-31-8(CAS DataBase Reference)
More
Less

Safety Information

Hazard Codes 
Xn
Risk Statements 
22
Safety Statements 
36
WGK Germany 
3
RTECS 
TZ1074800
Toxicity
LD50 in rats (mg/kg): 200 i.v., 750 orally (Morren)

MSDS

More
Less

Dropropizine Usage And Synthesis

Originator

Ribex,Formenti

Uses

antitussive

Uses

Dropropizine is a cough suppressant and central sedative therapeutic agent.

Definition

ChEBI: 3-(4-phenyl-1-piperazinyl)propane-1,2-diol is a member of piperazines.

Manufacturing Process

34 g 1,2-epoxy-3-hydroxypropane (glycide) in 50 ml of water were added to 64.8 g 1-phenylpiperazine in 80 ml of ethanol at the temperature not higher 50°C. The mixture was stood at night, then it was evaporated to dryness in vacuum and the stark product was recrystallized from 100 ml of acetone to give 60 g 1-phenyl-4-(2,3-dihydroxypropyl)piperazine (dropropizine) MP 105°C; BP 205°C/1 mm Hg.

Therapeutic Function

Antitussive

DropropizineSupplier

Shanghai YuanYe Biotechnology Co., Ltd. Gold
Tel
021-61312847; 18021002903
Email
3008007409@qq.com
J & K SCIENTIFIC LTD.
Tel
010-82848833 400-666-7788
Email
jkinfo@jkchemical.com
Meryer (Shanghai) Chemical Technology Co., Ltd.
Tel
021-61259108 18621169109
Email
market03@meryer.com
Energy Chemical
Tel
021-021-58432009 400-005-6266
Email
sales8178@energy-chemical.com
Shijiazhuang Sdyano Fine Chemical Co., Ltd.
Tel
0311-89250318 031166536426
Email
master@sjzsdyn.com