DELTORPHIN I
DELTORPHIN I Basic information
- Product Name:
- DELTORPHIN I
- Synonyms:
-
- DELTORPHIN I
- DELTORPHIN C
- DELTORPHIN 1
- [D-ALA2]DELTORPHIN I
- H-TYR-D-ALA-PHE-ASP-VAL-VAL-GLY-NH2
- TYR-D-ALA-PHE-ASP-VAL-VAL-GLY-NH2
- ala(2)-deltorphin
- tyr-D-ala-phe-asp-val-val-gly amide
- CAS:
- 122752-15-2
- MF:
- C37H52N8O10
- MW:
- 768.86
- Product Categories:
-
- Peptide
- Opioid receptor and opioid-like receptor
- Mol File:
- 122752-15-2.mol
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DELTORPHIN I Chemical Properties
- Boiling point:
- 1242.4±65.0 °C(Predicted)
- Density
- 1.284±0.06 g/cm3(Predicted)
- storage temp.
- -15°C
- solubility
- Soluble to 0.40 mg/ml in 50% acetonitrile / water
- pka
- 4.19±0.10(Predicted)
- form
- Powder
- color
- White to off-white
- Sequence
- Tyr-{d-Ala}-Phe-Asp-Val-Val-Gly-NH2
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DELTORPHIN I Usage And Synthesis
Uses
Selective delta-opioid receptor agonist
Definition
ChEBI: Deltorphin C is a peptide.
in vivo
Twice daily administration of Deltorphin I (20μg/mouse) for 4 days produces tolerance to Deltorphin I analgesia, as shown by the decrease in the analgesic response. The peak analgesic response to Deltorphin I (20 μg/mouse) at 10 min after injections is decreased from 8.36±0.28 s (the 1st day) to 4.53±0.14 s (the 4th day) markedly. Concurrent treatment of Melatonin (0.5, 1 and 2.5 mg/kg) and Deltorphin I (20 μg/mouse) twice daily for 4 days can attenuate the tolerance to Deltorphin I analgesia (P<0.05, <0.05 and <0.05), and this effect is dose dependent[1].
IC 50
δ Opioid Receptor/DOR
DELTORPHIN ISupplier
GL Biochem (Shanghai) Ltd
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- 21-61263452 13641803416
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Shanghai Hanhong Scientific Co.,Ltd.
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- 021-54306202 13764082696
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Chemsky（shanghai）International Co.,Ltd.
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- 021-50135380
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Cellmano Biotech Limited
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- 0551-65326643 18156095617
- info@cellmano.com
UHN Shanghai Research & Development Co., Ltd.
- Tel
- 021-58958002 18930822973
- sales@uhnshanghai.com
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DELTORPHIN I(122752-15-2)Related Product Information
- Boron triiodide
- Itd
- H-PHE-BETA-ALA-OH
- DELTORPHIN I
- Deltorphin [Met2]
- Dermenkephalin (Deltorphin, Dermorphin Gene-Associated Peptide, DGAP)
- deltorphin II, Ala(2)-,[D-Ala2,Glu4]deltorphin C,[D-Ala2,Glu4]Deltorphin II,DELTORPHIN B,DELTORPHIN II,[D-ALA2]-DELTORPHIN II
- deltorphin, Leu(2)-
- (MET2)-DELTORPHIN
- Deltorphin I (Deltorphin C)
- Deltorphin II [D-Ala2]
- DELTORPHIN A,DELTORPHIN,[D-Met2]deltorphin
- Deltorphin II (Deltorphin B)
- deltorphin, Ala(2)-Cys(4)-
- DELTORPHIN [D(ALA)2], BODIPY(R) 576/589
- deltorphin II, Ile(5,6)-
- DELTORPHIN II, (2-D-ALA), [TYROSYL-3,5-3H]-
- [D-Met6]deltorphin A