ChemicalBook > CAS DataBase List > Ralinepag

Ralinepag

Product Name
Ralinepag
CAS No.
1187856-49-0
Chemical Name
Ralinepag
Synonyms
APD811;APD-811;APD 811;Ralinepag;Sapanisertib;Ralinepag, 10 mM in DMSO;APD811;APD-811;APD 811;RALINEPAG;inhibit,APD-811,Ralinepag,Inhibitor,Prostaglandin Receptor,APD 811;2-((trans-4-((((4-Chlorophenyl)(phenyl)carbamoyl)oxy)methyl)cyclohexyl)methoxy)acetic acid;2-(((1R,4R)-4-((((4-CHLOROPHENYL)(PHENYL)CARBAMOYL)OXY)METHYL)CYCLOHEXYL)METHOXY)ACETIC ACID
CBNumber
CB03145551
Molecular Formula
C23H26ClNO5
Formula Weight
431.91
MOL File
1187856-49-0.mol
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Ralinepag Property

storage temp. 
Store at -20°C
solubility 
DMF: 15mg/mL; DMF:PBS (pH 7.2) (1:8): 0.11mg/mL; DMSO: 10mg/mL; Ethanol: 10mg/mL
form 
A solid
color 
White to off-white
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Hazard and Precautionary Statements (GHS)

Symbol(GHS)
Signal word
Warning
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N-Bromosuccinimide Price

Cayman Chemical
Product number
30009
Product name
Ralinepag
Packaging
1mg
Price
$37
Updated
2024/03/01
Cayman Chemical
Product number
30009
Product name
Ralinepag
Packaging
25mg
Price
$310
Updated
2024/03/01
Cayman Chemical
Product number
30009
Product name
Ralinepag
Packaging
5mg
Price
$134
Updated
2024/03/01
Cayman Chemical
Product number
30009
Product name
Ralinepag
Packaging
10mg
Price
$231
Updated
2024/03/01
TRC
Product number
R100095
Product name
Ralinepag
Packaging
2.5mg
Price
$605
Updated
2021/12/16
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Ralinepag Chemical Properties,Usage,Production

Uses

Ralinepag, is a potent non-prostanoid prostacyclin receptor agonist, with EC50s of 8.5 nM, 530 nM and 850 nM for human and rat IP receptor and human DP1 receptor, respectively.

in vivo

Ralinepag (30 mg/kg, p.o.) markedly reduces the monocrotaline (MCT)-induced increase in pulmonary arterial pressure and pulmonary vessel wall thickness in rats[1].

IC 50

hIP: 8.5 nM (EC50); rIP: 530 nM (EC50); hDP1: 850 nM (EC50)

Ralinepag Preparation Products And Raw materials

Raw materials

Preparation Products

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Ralinepag Suppliers

CHINA 47 United Kingdom 1 United States 6 Global 54
Shanghai Boyle Chemical Co., Ltd.
Tel
Fax
86-21-57758967
Email
sales@boylechem.com
Country
China
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2922
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Shanghai JiYi Biotechnology Co. Ltd.
Tel
13621943973
Fax
-
Email
sales@shjiyipharmatech.com
Country
China
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1166
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55
Shanghai Lollane Biological Technology Co.,Ltd.
Tel
021-52996696，15000506266 15000506266
Fax
+86-21-52996696
Country
China
ProdList
4827
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55
Shanghai EFE Biological Technology Co., Ltd.
Tel
021-65675885 18964387627
Fax
021-65675885
Email
info@efebio.com
Country
China
ProdList
9803
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58
Shanghai YuanYe Biotechnology Co., Ltd.
Tel
021-61312847; 18021002903
Fax
QQ:3008007432
Email
3008007409@qq.com
Country
China
ProdList
86249
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60
Shanghai Chaolan Chemical Technology Center
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021-QQ：65489617 15618227136
Fax
21-5161 9052
Email
Sales@ATKchemical.com
Country
China
ProdList
9532
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58
Amadis Chemical Company Limited
Tel
571-89925085
Fax
0086-571-89925065
Email
sales@amadischem.com
Country
China
ProdList
131957
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58
Lynnchem
Tel
86-(0)29-85992781 17792393971
Email
info@lynnchem.com
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China
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58
Novachemistry
Tel
44-20819178-90 02081917890
Fax
(0)2080432064
Email
info@novachemistry.com
Country
United Kingdom
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4381
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58
Shanghai Biopharmaleader Co., Ltd.
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+86 18721201413
Fax
+86 (21) 5775-8967
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sales@biopharmaleader.com
Country
China
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1720
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1187856-49-0, RalinepagRelated Search:


  • Ralinepag
  • Sapanisertib
  • 2-(((1R,4R)-4-((((4-CHLOROPHENYL)(PHENYL)CARBAMOYL)OXY)METHYL)CYCLOHEXYL)METHOXY)ACETIC ACID
  • APD 811
  • APD811
  • APD-811
  • APD811;APD-811;APD 811;RALINEPAG
  • Acetic acid, 2-[[trans-4-[[[[(4-chlorophenyl)phenylamino]carbonyl]oxy]methyl]cyclohexyl]methoxy]-
  • inhibit,APD-811,Ralinepag,Inhibitor,Prostaglandin Receptor,APD 811
  • 2-((trans-4-((((4-Chlorophenyl)(phenyl)carbamoyl)oxy)methyl)cyclohexyl)methoxy)acetic acid
  • Ralinepag, 10 mM in DMSO
  • 1187856-49-0