ChemicalBook > CAS DataBase List > MMSET-IN-1
MMSET-IN-1
- Product Name
- MMSET-IN-1
- CAS No.
- 1998139-29-9
- Chemical Name
- MMSET-IN-1
- Synonyms
- MMSET-IN-1;MMSETIN1,MMSET IN 1;β-D-allo-Decofuranuronic acid, 9-amino-1-(6-amino-9H-purin-9-yl)-1,5,6,7,8,9-hexadeoxy-6-(propylamino)-, (6ξ)-
- CBNumber
- CB04668215
- Molecular Formula
- C18H29N7O5
- Formula Weight
- 423.47
- MOL File
- 1998139-29-9.mol
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MMSET-IN-1 Property
- Boiling point:
- 753.8±70.0 °C(Predicted)
- Density
- 1.66±0.1 g/cm3(Predicted)
- storage temp.
- Store at -20°C
- solubility
- Soluble in DMSO
- pka
- 2.47±0.28(Predicted)
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MMSET-IN-1 Chemical Properties,Usage,Production
Description
MMSET-IN-1 is a multiple myeloma SET domain (MMSET, aka NSD2/WHSC1) inhibitor against SETD2 and MMSET with IC50s of 0.49 and 3.3 μM, respectively. MMSET-IN-1 has a Kd of 1.6 μM for MMSET[1]. IC50: 0.49 μM (SETD2), 3.3 μM (MMSET)[1]Kd: 1.6 μM[1]
References
[1]. Tisi D, et al. Structure of the Epigenetic Oncogene MMSET and Inhibition by N-Alkyl Sinefungin Derivatives. ACS Chem Biol. 2016 Nov 18;11(11):3093-3105.
MMSET-IN-1 Preparation Products And Raw materials
Raw materials
Preparation Products
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MMSET-IN-1 Suppliers
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