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Z-Val-Arg-Pro-DL-Arg-fluoromethylketone trifluoroacetate salt

Product Name
Z-Val-Arg-Pro-DL-Arg-fluoromethylketone trifluoroacetate salt
CAS No.
1926163-57-6
Chemical Name
Z-Val-Arg-Pro-DL-Arg-fluoromethylketone trifluoroacetate salt
Synonyms
Z-VRPR-FMK trifluoroacetate;Z-Val-Arg-Pro-DL-Arg-fluoromethylketone trifluoroacetate salt;L-Prolinamide, N-[(phenylmethoxy)carbonyl]-L-valyl-L-arginyl-N-[4-[(aminoiminomethyl)amino]-1-(2-fluoroacetyl)butyl]-
CBNumber
CB04915751
Molecular Formula
C31H49FN10O6
Formula Weight
676.78
MOL File
1926163-57-6.mol
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Z-Val-Arg-Pro-DL-Arg-fluoromethylketone trifluoroacetate salt Property

Density 
1.38±0.1 g/cm3(Predicted)
pka
11.06±0.46(Predicted)
Sequence
Z-Val-Arg-Pro-{DL-Arg}-{Fluoromethylketone}
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Hazard and Precautionary Statements (GHS)

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N-Bromosuccinimide Price

Chem-Impex
Product number
32776
Product name
Z-Val-Arg-Pro-DL-Arg-fluoromethylketone trifluoroacetate salt
Packaging
500MG
Price
$310.5
Updated
2021/12/16
Chem-Impex
Product number
32776
Product name
Z-Val-Arg-Pro-DL-Arg-fluoromethylketone trifluoroacetate salt
Packaging
1MG
Price
$550
Updated
2021/12/16
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Z-Val-Arg-Pro-DL-Arg-fluoromethylketone trifluoroacetate salt Chemical Properties,Usage,Production

Uses

Z-Val-Arg-Pro-DL-Arg-Fluoromethylketone is a potent MALT1 inhibitor. Z-Val-Arg-Pro-DL-Arg-Fluoromethylketone inhibits cell proliferation and migration. Z-Val-Arg-Pro-DL-Arg-Fluoromethylketone shows anticancer activity[1].

in vivo

Z-Val-Arg-Pro-DL-Arg-Fluoromethylketone (37.5 M*0.2 mL; every other day for 12 days) inhibits the growth of the tumor in mouse[1].

Animal Model:4-6 weeks, 16-20 g, Female BALB/c nude mice (OCI-LY10 cells)[1]
Dosage:37.5 M*0.2 mL
Administration:Every other day for 12 days
Result:Inhibited the growth of the xenografts and decreased the expression of P65.

References

[1] Feng J, et al. Z-VRPR-FMK can inhibit the growth and invasiveness of diffuse large B-cell lymphoma by depressing NF-κB activation and MMP expression induced by MALT1. Int J Clin Exp Pathol. 2019 Jun 1;12(6):1947-1955. PMID:31934017

Z-Val-Arg-Pro-DL-Arg-fluoromethylketone trifluoroacetate salt Preparation Products And Raw materials

Raw materials

Preparation Products

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Z-Val-Arg-Pro-DL-Arg-fluoromethylketone trifluoroacetate salt Suppliers

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1926163-57-6, Z-Val-Arg-Pro-DL-Arg-fluoromethylketone trifluoroacetate saltRelated Search:


  • Z-Val-Arg-Pro-DL-Arg-fluoromethylketone trifluoroacetate salt
  • L-Prolinamide, N-[(phenylmethoxy)carbonyl]-L-valyl-L-arginyl-N-[4-[(aminoiminomethyl)amino]-1-(2-fluoroacetyl)butyl]-
  • Z-VRPR-FMK trifluoroacetate
  • 1926163-57-6
  • C31H49FN10O6