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E3 ligase Ligand-Linker Conjugates 38

Product Name
E3 ligase Ligand-Linker Conjugates 38
CAS No.
2095244-52-1
Chemical Name
E3 ligase Ligand-Linker Conjugates 38
Synonyms
cIAP1 Ligand-Linker Conjugates 12;E3 ligase Ligand-Linker Conjugates 38;tert-butyl N-[(1S)-1-{[(1S)-1-cyclohexyl-2-[(2S)-2-[4-(3-{2-[2-(2-{2-[(4-methylbenzenesulfonyl)oxy]ethoxy}ethoxy)ethoxy]ethoxy}benzoyl)-1,3-thiazol-2-yl]pyrrolidin-1-yl]-2-oxoethyl]carbamoyl}ethyl]-N-methylcarbamate;Benzenesulfonic acid, 4-methyl-, 2-[2-[2-[2-[3-[[2-[(2S)-1-[(2S)-2-cyclohexyl-2-[[(2S)-2-[[(1,1-dimethylethoxy)carbonyl]methylamino]-1-oxopropyl]amino]acetyl]-2-pyrrolidinyl]-4-thiazolyl]carbonyl]phenoxy]ethoxy]ethoxy]ethoxy]ethyl ester
CBNumber
CB08054715
Molecular Formula
C46H64N4O12S2
Formula Weight
929.15
MOL File
2095244-52-1.mol
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E3 ligase Ligand-Linker Conjugates 38 Property

Boiling point:
999.9±65.0 °C(Predicted)
Density 
1.239±0.06 g/cm3(Predicted)
pka
14.02±0.46(Predicted)
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Hazard and Precautionary Statements (GHS)

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E3 ligase Ligand-Linker Conjugates 38 Chemical Properties,Usage,Production

Uses

cIAP1 Ligand-Linker Conjugates 12 incorporates an IAP ligand for the E3 ubiquitin ligase, and a PROTAC linker. cIAP1 Ligand-Linker Conjugates 12 can be used to design SNIPERs[1].

IC 50

cIAP1

References

[1] Ohoka N, et al. In Vivo Knockdown of Pathogenic Proteins via Specific and Nongenetic Inhibitor of Apoptosis Protein (IAP)-dependent Protein Erasers (SNIPERs). J Biol Chem. 2017 Mar 17;292(11):4556-4570. DOI:10.1074/jbc.M116.768853

E3 ligase Ligand-Linker Conjugates 38 Preparation Products And Raw materials

Raw materials

Preparation Products

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E3 ligase Ligand-Linker Conjugates 38 Suppliers

Jilin Province Woda Biotechnology Co., Ltd.
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2095244-52-1, E3 ligase Ligand-Linker Conjugates 38Related Search:


  • cIAP1 Ligand-Linker Conjugates 12
  • E3 ligase Ligand-Linker Conjugates 38
  • Benzenesulfonic acid, 4-methyl-, 2-[2-[2-[2-[3-[[2-[(2S)-1-[(2S)-2-cyclohexyl-2-[[(2S)-2-[[(1,1-dimethylethoxy)carbonyl]methylamino]-1-oxopropyl]amino]acetyl]-2-pyrrolidinyl]-4-thiazolyl]carbonyl]phenoxy]ethoxy]ethoxy]ethoxy]ethyl ester
  • tert-butyl N-[(1S)-1-{[(1S)-1-cyclohexyl-2-[(2S)-2-[4-(3-{2-[2-(2-{2-[(4-methylbenzenesulfonyl)oxy]ethoxy}ethoxy)ethoxy]ethoxy}benzoyl)-1,3-thiazol-2-yl]pyrrolidin-1-yl]-2-oxoethyl]carbamoyl}ethyl]-N-methylcarbamate
  • 2095244-52-1