perlapine
- Product Name
- perlapine
- CAS No.
- 1977-11-3
- Chemical Name
- perlapine
- Synonyms
- HF 2333;Hypnodin;AW 14-2333;6-(4-Methyl-1-piperazinyl)-11H-dibenz[b,e]azepin;6-(4-Methyl-1-piperazinyl)-11H-dibenz[b,e]azepine;11H-Dibenz[b,e]azepine, 6-(4-methyl-1-piperazinyl)-;6-(4-methylpiperazin-1-yl)-11H-benzo[c][1]benzazepine
- CBNumber
- CB11388928
- Molecular Formula
- C19H21N3
- Formula Weight
- 291.39
- MOL File
- 1977-11-3.mol
perlapine Property
- Melting point:
- 136-138°
- Boiling point:
- 423.4°C (rough estimate)
- Density
- 1.0521 (rough estimate)
- refractive index
- 1.6080 (estimate)
- storage temp.
- Store at -20°C
- solubility
- DMF: 10 mg/ml; DMSO: 10 mg/ml; DMSO:PBS (pH 7.2) (1:1): 0.5 mg/ml; Ethanol: 5 mg/ml
- form
- A crystalline solid
- pka
- 8.00±0.20(Predicted)
- color
- White
Safety
- Toxicity
- LD50 in male, female mice, rats (mg/kg): 61, 61, 60, 66 i.v.; 250, 300, 480, 420 s.c., 270, 280, 660, 720 orally (Yokotani)
Hazard and Precautionary Statements (GHS)
- Symbol(GHS)
-
- Signal word
- Warning
- Hazard statements
-
H302Harmful if swallowed
- Precautionary statements
-
P264Wash hands thoroughly after handling.
P264Wash skin thouroughly after handling.
P270Do not eat, drink or smoke when using this product.
P301+P312IF SWALLOWED: call a POISON CENTER or doctor/physician IF you feel unwell.
P330Rinse mouth.
P501Dispose of contents/container to..…
N-Bromosuccinimide Price
- Product number
- 17756
- Product name
- Perlapine
- Purity
- ≥98%
- Packaging
- 1mg
- Price
- $57
- Updated
- 2024/03/01
- Product number
- 17756
- Product name
- Perlapine
- Purity
- ≥98%
- Packaging
- 5mg
- Price
- $117
- Updated
- 2024/03/01
- Product number
- 17756
- Product name
- Perlapine
- Purity
- ≥98%
- Packaging
- 10mg
- Price
- $172
- Updated
- 2024/03/01
- Product number
- N900420
- Product name
- Perlapine
- Packaging
- 10mg
- Price
- $135
- Updated
- 2021/12/16
- Product number
- API0003796
- Product name
- PERLAPINE
- Purity
- 95.00%
- Packaging
- 20MG
- Price
- $238
- Updated
- 2021/12/16
perlapine Chemical Properties,Usage,Production
Uses
Perlapine is an atypical neuroleptic that blocks dopamine and serotonin (5-HT) receptors (Kis = 60, 30, and 30 nM for D2, D4, and 5-HT2A, respectively). Perlapine is also an agonist for hM3Dq, a designer receptor exclusively activated by designer drugs (DREADD) derived from the human muscarinic acetylcholine M3 receptor that activates neuronal firing. Perlapine displays >10,000-fold selectivity for hM3Dq over hM3.
Uses
Perlapine exhibits antipsychotic activity and blocks dopamine and serotonin receptors. Perlapine is also a novel agonist of hM3Dq, a designer receptor exclusively activated by designer drugs (DREADD).
Definition
ChEBI: Perlapine is an organic molecular entity.
storage
Room temperature
perlapine Preparation Products And Raw materials
Raw materials
Preparation Products
perlapine Suppliers
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