perlapine

Product Name: perlapine
CAS No.: 1977-11-3
Chemical Name: perlapine
Synonyms: HF 2333;Hypnodin;AW 14-2333;6-(4-Methyl-1-piperazinyl)-11H-dibenz[b,e]azepin;6-(4-Methyl-1-piperazinyl)-11H-dibenz[b,e]azepine;11H-Dibenz[b,e]azepine, 6-(4-methyl-1-piperazinyl)-;6-(4-methylpiperazin-1-yl)-11H-benzo[c][1]benzazepine
CBNumber: CB11388928
Molecular Formula: C19H21N3
Formula Weight: 291.39
MOL File: 1977-11-3.mol

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perlapine Property

Melting point:: 136-138°
Boiling point:: 423.4°C (rough estimate)
Density: 1.0521 (rough estimate)
refractive index: 1.6080 (estimate)
storage temp.: Store at -20°C
solubility: DMF: 10 mg/ml; DMSO: 10 mg/ml; DMSO:PBS (pH 7.2) (1:1): 0.5 mg/ml; Ethanol: 5 mg/ml
form: A crystalline solid
pka: 8.00±0.20(Predicted)
color: White

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Safety

Toxicity: LD50 in male, female mice, rats (mg/kg): 61, 61, 60, 66 i.v.; 250, 300, 480, 420 s.c., 270, 280, 660, 720 orally (Yokotani)

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Hazard and Precautionary Statements (GHS)

Symbol(GHS)

Signal word

Warning

Hazard statements

H302Harmful if swallowed

Precautionary statements

P264Wash hands thoroughly after handling.

P264Wash skin thouroughly after handling.

P270Do not eat, drink or smoke when using this product.

P301+P312IF SWALLOWED: call a POISON CENTER or doctor/physician IF you feel unwell.

P330Rinse mouth.

P501Dispose of contents/container to..…

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N-Bromosuccinimide Price

Cayman Chemical

Product number: 17756
Product name: Perlapine
Purity: ≥98%
Packaging: 1mg
Price: $57
Updated: 2024/03/01

Cayman Chemical

Product number: 17756
Product name: Perlapine
Purity: ≥98%
Packaging: 5mg
Price: $117
Updated: 2024/03/01

Cayman Chemical

Product number: 17756
Product name: Perlapine
Purity: ≥98%
Packaging: 10mg
Price: $172
Updated: 2024/03/01

TRC

Product number: N900420
Product name: Perlapine
Packaging: 10mg
Price: $135
Updated: 2021/12/16

American Custom Chemicals Corporation

Product number: API0003796
Product name: PERLAPINE
Purity: 95.00%
Packaging: 20MG
Price: $238
Updated: 2021/12/16

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perlapine Chemical Properties,Usage,Production

Uses

Perlapine is an atypical neuroleptic that blocks dopamine and serotonin (5-HT) receptors (Kis = 60, 30, and 30 nM for D2, D4, and 5-HT2A, respectively). Perlapine is also an agonist for hM3Dq, a designer receptor exclusively activated by designer drugs (DREADD) derived from the human muscarinic acetylcholine M3 receptor that activates neuronal firing. Perlapine displays >10,000-fold selectivity for hM3Dq over hM3.

Uses

Perlapine exhibits antipsychotic activity and blocks dopamine and serotonin receptors. Perlapine is also a novel agonist of hM3Dq, a designer receptor exclusively activated by designer drugs (DREADD).

Definition

ChEBI: Perlapine is an organic molecular entity.

storage

Room temperature

perlapine Preparation Products And Raw materials

Raw materials

Preparation Products

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perlapine Suppliers

China 11 South Korea 1 United Kingdom 1 United States 3 Global 16

TargetMol Chemicals Inc.

Tel: +1-781-999-5354 +1-00000000000
Email: marketing@targetmol.com
Country: United States
ProdList: 32165
Advantage: 58

HANGZHOU CLAP TECHNOLOGY CO.,LTD

Tel: 86-571-88216897,88216896 13588875226
Fax: 86-571-88216895
Email: sales@hzclap.com
Country: CHINA
ProdList: 6312
Advantage: 58

ChemeGen(Shanghai) Biotechnology Co.,Ltd.

Tel: 18818260767
Fax: QQ 3610331285
Email: sales@chemegen.com
Country: China
ProdList: 11217
Advantage: 58

Guangzhou Younan Technology Co., Ltd

Tel: 020-82000279 18988968278
Fax: QQ：3283937693
Email: sales@ubiochem.com
Country: China
ProdList: 4297
Advantage: 58

Energy Chemical

Tel: 021-58432009 400-005-6266
Fax: 021-58436166
Email: marketing1@energy-chemical.com
Country: China
ProdList: 44808
Advantage: 58

MedBioPharmaceutical Technology Inc

Tel: 021-69568360 18916172912
Email: order@med-bio.cn
Country: China
ProdList: 8140
Advantage: 58

TargetMol Chemicals Inc.

Tel: 4008200310
Email: marketing@tsbiochem.com
Country: China
ProdList: 24647
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Shanghai Yifei Biotechnology Co. , Ltd.

Tel: 021-65675885 18964387627
Email: customer_service@efebio.com
Country: China
ProdList: 11974
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RD International Technology Co., Limited

Tel: 18024082417
Email: market@ubiochem.com
Country: China
ProdList: 9272
Advantage: 58

TargetMol Chemicals Inc.

Tel
Email: support@targetmol.com
Country: United States
ProdList: 38632
Advantage: 58

1977-11-3, perlapineRelated Search:

FLUPERLAPINE 2-ETHYL-BENZAMIDINE perlapine 1-(2-METHYLBENZYL)PIPERAZINE

6-(4-Methyl-1-piperazinyl)-11H-dibenz[b,e]azepin

AW 14-2333

HF 2333

Hypnodin

6-(4-methylpiperazin-1-yl)-11H-benzo[c][1]benzazepine

6-(4-Methyl-1-piperazinyl)-11H-dibenz[b,e]azepine

11H-Dibenz[b,e]azepine, 6-(4-methyl-1-piperazinyl)-

1977-11-3