(AR)-A-CYCLOPENTYL-A-HYDROXY-N-[1-(4-METHYL-3-PENTENYL)-4-PIPERIDINYL]BENZENEACETAMIDE FUMARATE

Product Name: (AR)-A-CYCLOPENTYL-A-HYDROXY-N-[1-(4-METHYL-3-PENTENYL)-4-PIPERIDINYL]BENZENEACETAMIDE FUMARATE
CAS No.: 244277-89-2
Chemical Name: (AR)-A-CYCLOPENTYL-A-HYDROXY-N-[1-(4-METHYL-3-PENTENYL)-4-PIPERIDINYL]BENZENEACETAMIDE FUMARATE
Synonyms: J 104129 FUMARATE;Benzeneacetamide, α-cyclopentyl-α-hydroxy-N-[1-(4-methyl-3-penten-1-yl)-4-piperidinyl]-, (αR)-;(αR)-α-Cyclopentyl-α-hydroxy-N-[1-(4-methyl-3-pentenyl)-4-piperidinyl]benzeneacetamidefumarate;(AR)-A-CYCLOPENTYL-A-HYDROXY-N-[1-(4-METHYL-3-PENTENYL)-4-PIPERIDINYL]BENZENEACETAMIDE FUMARATE
CBNumber: CB12450341
Molecular Formula: C24H36N2O2
Formula Weight: 384.55
MOL File: 244277-89-2.mol

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(AR)-A-CYCLOPENTYL-A-HYDROXY-N-[1-(4-METHYL-3-PENTENYL)-4-PIPERIDINYL]BENZENEACETAMIDE FUMARATE Property

storage temp.: Store at +4°C
solubility: <50.06mg/ml in DMSO; <25.03mg/ml in ethanol

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Hazard and Precautionary Statements (GHS)

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N-Bromosuccinimide Price

Tocris

Product number: 2507
Product name: J104129fumarate
Purity: ≥99%(HPLC)
Packaging: 10
Price: $217
Updated: 2021/12/16

Usbiological

Product number: 255545
Product name: J 104129 Fumarate
Packaging: 10mg
Price: $480
Updated: 2021/12/16

TRC

Product number: J211990
Product name: J104129
Packaging: 10mg
Price: $160
Updated: 2021/12/16

American Custom Chemicals Corporation

Product number: API0019220
Product name: (ALPHA-R)-ALPHA-CYCLOPENTYL-ALPHA-HYDROXY-N-[1-(4-METHYL-3-PENTENYL)-4-PIPERIDINYL]BENZENEACETAMIDE FUMARATE
Purity: 95.00%
Packaging: 5MG
Price: $500.62
Updated: 2021/12/16

ApexBio Technology

Product number: B7083
Product name: J104129fumarate
Packaging: 10mg
Price: $322
Updated: 2021/12/16

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(AR)-A-CYCLOPENTYL-A-HYDROXY-N-[1-(4-METHYL-3-PENTENYL)-4-PIPERIDINYL]BENZENEACETAMIDE FUMARATE Chemical Properties,Usage,Production

Uses

J 104129 is a mAChR M3 antagonist.

Biological Activity

Potent M 3 muscarinic receptor antagonist that displays ~ 120-fold selectivity over M 2 receptors (K i values are 4.2, 19 and 490 nM for human M 3 , M 1 and M 2 receptors respectively). Exhibits > 250-fold bronchial selectivity; inhibits ACh-induced bronchoconstriction but not ACh-induced bradycardia (K B values are 3.3 and 170 nM for rat trachea M 3 and rat right atria M 2 receptors respectively).

(AR)-A-CYCLOPENTYL-A-HYDROXY-N-[1-(4-METHYL-3-PENTENYL)-4-PIPERIDINYL]BENZENEACETAMIDE FUMARATE Preparation Products And Raw materials

Raw materials

Preparation Products

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(AR)-A-CYCLOPENTYL-A-HYDROXY-N-[1-(4-METHYL-3-PENTENYL)-4-PIPERIDINYL]BENZENEACETAMIDE FUMARATE Suppliers

China 7 United Kingdom 1 United States 6 Global 14

Tocris Bioscience

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244277-89-2, (AR)-A-CYCLOPENTYL-A-HYDROXY-N-[1-(4-METHYL-3-PENTENYL)-4-PIPERIDINYL]BENZENEACETAMIDE FUMARATERelated Search:

(2-CYCLOPENTYL-2-PHENYLETHYL)AMINE (AR)-A-CYCLOPENTYL-A-HYDROXY-N-[1-(4-METHYL-3-PENTENYL)-4-PIPERIDINYL]BENZENEACETAMIDE FUMARATE

(AR)-A-CYCLOPENTYL-A-HYDROXY-N-[1-(4-METHYL-3-PENTENYL)-4-PIPERIDINYL]BENZENEACETAMIDE FUMARATE

J 104129 FUMARATE

(αR)-α-Cyclopentyl-α-hydroxy-N-[1-(4-methyl-3-pentenyl)-4-piperidinyl]benzeneacetamidefumarate

Benzeneacetamide, α-cyclopentyl-α-hydroxy-N-[1-(4-methyl-3-penten-1-yl)-4-piperidinyl]-, (αR)-

244277-89-2

C24H36N2O2C4H4O4