ChemicalBook > CAS DataBase List > (+)-JQ1 PA

(+)-JQ1 PA

Product Name
(+)-JQ1 PA
CAS No.
2115701-93-2
Chemical Name
(+)-JQ1 PA
Synonyms
(+)-JQ1 PA;PubChem ID: 134821687;JQ1 PA;JQ-1 PA;JQ 1 PA;inhibit,(+) JQ1 PA,(+)-JQ1 PA,Inhibitor,Epigenetic Reader Domain,(+)JQ1 PA,(+)-JQ-1 PA;(6S)-4-(4-Chlorophenyl)-2,3,9-trimethyl-N-2-propyn-1-yl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetamide;6H-Thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetamide, 4-(4-chlorophenyl)-2,3,9-trimethyl-N-2-propyn-1-yl-, (6S)-;(S)-2-(4-(4-Chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl)-N-(prop-2-yn-1-yl)acetamide
CBNumber
CB14718443
Molecular Formula
C22H20ClN5OS
Formula Weight
437.95
MOL File
2115701-93-2.mol
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(+)-JQ1 PA Property

storage temp. 
Store at -20°C
solubility 
DMF: 30 mg/ml; DMSO: 30 mg/ml; DMSO:PBS (pH 7.2) (1:6): 0.14 mg/ml; Ethanol: 25 mg/ml
form 
A crystalline solid
color 
Light yellow to yellow
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Hazard and Precautionary Statements (GHS)

Symbol(GHS)
Signal word
Warning
Hazard statements

H302Harmful if swallowed

H315Causes skin irritation

H319Causes serious eye irritation

H335May cause respiratory irritation

Precautionary statements

P261Avoid breathing dust/fume/gas/mist/vapours/spray.

P280Wear protective gloves/protective clothing/eye protection/face protection.

P301+P312IF SWALLOWED: call a POISON CENTER or doctor/physician IF you feel unwell.

P302+P352IF ON SKIN: wash with plenty of soap and water.

P305+P351+P338IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses, if present and easy to do. Continuerinsing.

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N-Bromosuccinimide Price

Cayman Chemical
Product number
30414
Product name
(+)-JQ1 PA
Packaging
1mg
Price
$32
Updated
2024/03/01
Cayman Chemical
Product number
30414
Product name
(+)-JQ1 PA
Packaging
25mg
Price
$533
Updated
2024/03/01
Cayman Chemical
Product number
30414
Product name
(+)-JQ1 PA
Packaging
5mg
Price
$139
Updated
2024/03/01
Cayman Chemical
Product number
30414
Product name
(+)-JQ1 PA
Packaging
10mg
Price
$243
Updated
2024/03/01
Tocris
Product number
6589
Product name
(+)-JQ1PA
Purity
≥95%(HPLC)
Packaging
25
Price
$482
Updated
2021/12/16
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(+)-JQ1 PA Chemical Properties,Usage,Production

Biological Activity

(+)-JQ1 PA is a derivative of the bromodomain and extra terminal domain (BET) inhibitor JQ1 with an IC50 value of 10.4 nM.

in vitro

(+)-JQ1 PA is a derivative of JQ1, which is the inhibitor of BET. The IC 50 of (+)-JQ1 PA for BET is 10.4 nM, and the IC 50 of JQ1 is 14.3 nM in MV4;11 cells.

target

10.4 nM (BET).

storage

Store at -20°C

(+)-JQ1 PA Preparation Products And Raw materials

Raw materials

Preparation Products

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(+)-JQ1 PA Suppliers

China 33 United Kingdom 1 United States 5 Global 39
Tocris Bioscience
Tel
--
Fax
--
Email
customerservice@tocris.co.uk
Country
United Kingdom
ProdList
5726
Advantage
77

2115701-93-2, (+)-JQ1 PARelated Search:


  • (+)-JQ1 PA
  • JQ1 PA;JQ-1 PA;JQ 1 PA
  • (6S)-4-(4-Chlorophenyl)-2,3,9-trimethyl-N-2-propyn-1-yl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetamide
  • PubChem ID: 134821687
  • 6H-Thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetamide, 4-(4-chlorophenyl)-2,3,9-trimethyl-N-2-propyn-1-yl-, (6S)-
  • inhibit,(+) JQ1 PA,(+)-JQ1 PA,Inhibitor,Epigenetic Reader Domain,(+)JQ1 PA,(+)-JQ-1 PA
  • (S)-2-(4-(4-Chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl)-N-(prop-2-yn-1-yl)acetamide
  • 2115701-93-2