5-METHOXY-6-AZAINDOLE
- Product Name
- 5-METHOXY-6-AZAINDOLE
- CAS No.
- 17288-53-8
- Chemical Name
- 5-METHOXY-6-AZAINDOLE
- Synonyms
- 5-Methxy-6-azaindole;5-METHOXY-6-AZAINDOLE;5-Methoxy-6-azaindole 96%;5-Methyl-1H-pyrrolo[2,3-c]pyridine;5-Methoxy-1H-pyrrolo[2,3-c]pyridine;5-Metho×y-1H-pyrrolo[2,3-c]pyridine;1H-Pyrrolo[2,3-c]pyridine, 5-Methoxy-
- CBNumber
- CB1841543
- Molecular Formula
- C8H8N2O
- Formula Weight
- 148.16
- MOL File
- 17288-53-8.mol
5-METHOXY-6-AZAINDOLE Property
- Melting point:
- 122-127 °C
- Boiling point:
- 304℃
- Density
- 1.244
- Flash point:
- 105℃
- storage temp.
- 2-8°C
- pka
- 14.36±0.40(Predicted)
- form
- powder
- Appearance
- Off-white to gray Solid
Hazard and Precautionary Statements (GHS)
- Symbol(GHS)
-
- Signal word
- Warning
- Hazard statements
-
H302Harmful if swallowed
- Precautionary statements
-
P280Wear protective gloves/protective clothing/eye protection/face protection.
P305+P351+P338IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses, if present and easy to do. Continuerinsing.
N-Bromosuccinimide Price
- Product number
- 696463
- Product name
- 5-Methoxy-6-azaindole
- Purity
- 96%
- Packaging
- 1g
- Price
- $658.7
- Updated
- 2025/07/31
- Product number
- M269475
- Product name
- 5-Methoxy-1H-pyrrolo[2,3-c]pyridine
- Packaging
- 50mg
- Price
- $45
- Updated
- 2021/12/16
- Product number
- M269475
- Product name
- 5-Methoxy-1H-pyrrolo[2,3-c]pyridine
- Packaging
- 100mg
- Price
- $60
- Updated
- 2021/12/16
- Product number
- M269475
- Product name
- 5-Methoxy-1H-pyrrolo[2,3-c]pyridine
- Packaging
- 500mg
- Price
- $130
- Updated
- 2021/12/16
- Product number
- 4H56-1-609
- Product name
- 5-Methoxy-6-azaindole
- Packaging
- 1g
- Price
- $375
- Updated
- 2021/12/16
5-METHOXY-6-AZAINDOLE Chemical Properties,Usage,Production
Uses
Reactant for preparation of indole sulfonamides as HIV entry inhibitors1Reactant for synthesis of melatoninergic ligands including azaindole moiety2
Uses
Reactant for preparation of indole sulfonamides as HIV entry inhibitors
Reactant for synthesis of melatoninergic ligands including azaindole moiety
Synthesis
21901-41-7
23056-33-9
17288-53-8
Example 12: Synthesis of 5-methoxypyrrolo[2,3-c]pyridine (Compound 9) 4-Methyl-5-nitro-1H-pyridin-2-one (5.00 g, 32.44 mmol) was mixed with thionyl chloride (20 ml), two drops of dimethylformamide were added under nitrogen protection and heated to reflux for 52 hours. Upon completion of the reaction, the resulting orange solution was concentrated under reduced pressure, added a small amount of anhydrous toluene and concentrated again under reduced pressure to remove residual thionyl chloride. Subsequently, the crude product was purified by column chromatography on silica gel (silica gel was pre-dried overnight at 150 °C under vacuum, about 100 g), and the eluent was dichloromethane (11). The eluate was collected and concentrated under reduced pressure to afford 2-chloro-4-methyl-5-nitropyridine (5.30 g, 30.71 mmol, 95% yield) as an orange oil, which could be crystallized by cooling to below 0 °C. Product characterization data. IR (CHCl3): 1605, 1550, 1520, 1450, 1360, 1345 cm-1;. 1H NMR (CDCl3): δ 9.03 (s, 1H), 7.83 (s, 1H), 2.60 (s, 3H); δ 2.60 (s, 3H). LRMS (m/z, relative intensity): 174 (25), 173 (19), 172 (M+, 68), 157 (74), 155 (100), 128 (27), 101 (47), 100 (55), 99 (74), 90 (43), 75 (36).
References
[1] Patent: US5051412, 1991, A
5-METHOXY-6-AZAINDOLE Preparation Products And Raw materials
Raw materials
Preparation Products
5-METHOXY-6-AZAINDOLE Suppliers
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View Lastest Price from 5-METHOXY-6-AZAINDOLE manufacturers
- Product
- 5-METHOXY-6-AZAINDOLE 17288-53-8
- Price
- US $9.80/KG
- Min. Order
- 1g
- Purity
- ≥99%
- Supply Ability
- 100kg
- Release date
- 2020-01-08