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Deslorelin acetate

Product Name
Deslorelin acetate
CAS No.
82318-06-7
Chemical Name
Deslorelin acetate
Synonyms
H 4065 Acetate;SoMagard Aceta;PTL 3001 Acetate;BacheM 9022 Acetate;D-Trp LHRH-PEA Acetate;Deslorelin Acetate(acetate);D-Trp6-Pro9-N-ethylaMide-LH-RH Acetate;6-D-Tryptophan-9-(N-ethyl-L-prolinaMide)-1-9-luteinizing HorMone-releasing Factor (Swine) Monoacetate
CBNumber
CB21105098
Molecular Formula
C66H87N17O14
Formula Weight
1342.50248
MOL File
82318-06-7.mol
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Hazard and Precautionary Statements (GHS)

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N-Bromosuccinimide Price

Biosynth Carbosynth
Product number
FD21216
Product name
Deslorelin
Packaging
50mg
Price
$65
Updated
2021/12/16
Biosynth Carbosynth
Product number
FD21216
Product name
Deslorelin
Packaging
100mg
Price
$100
Updated
2021/12/16
Biosynth Carbosynth
Product number
FD21216
Product name
Deslorelin
Packaging
250mg
Price
$200
Updated
2021/12/16
Biosynth Carbosynth
Product number
FD21216
Product name
Deslorelin
Packaging
500mg
Price
$320
Updated
2021/12/16
Biosynth Carbosynth
Product number
FD21216
Product name
Deslorelin
Packaging
1g
Price
$510
Updated
2021/12/16
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Deslorelin acetate Chemical Properties,Usage,Production

Description

Deslorelin Acetate is a synthetic nonapeptide analogue of the natural gonadotrophin releasing hormone (GnRH) with potential antineoplastic activity. Deslorelin binds to and activates pituitary gonadotropin releasing hormone (GnRH) receptors. Continuous, prolonged administration of goserelin in males results in pituitary GnRH receptor desensitization and inhibition of pituitary secretion of follicle stimulating hormone (FSH) and luteinizing hormone (LH), leading to a significant decline in testosterone production; in females, prolonged administration results in a decrease in estradiol production.

Uses

Deslorelin acetate is an injectable gonadotropin-releasing hormone (GnRH) super-agonist (also known as an LHRH agonist), used in treatment of precocious puberty and commonly used in veterinary medicine to induce ovulation in mares.

Preparation

Deslorelin acetate is synthesized from the corresponding protected amino acid monomers by solid or liquid phase synthesis.

References

[1] C L ACKERMANN. Ovarian activity reversibility after the use of deslorelin acetate as a short-term contraceptive in domestic queens.[J]. Theriogenology, 2012, 78 4: 817-822. DOI:10.1016/j.theriogenology.2012.03.030.
[2] R. NOVOTNY . Reversible suppression of sexual activity in tomcats with deslorelin implant[J]. Theriogenology, 2012, 78 4: Pages 848-857. DOI:10.1016/j.theriogenology.2012.03.035.
[3] Y CETIN. Long-term effect of deslorelin implant on ovarian pre-antral follicles and uterine histology in female rats.[J]. Reproduction in Domestic Animals, 2013, 48 2: 195-199. DOI:10.1111/j.1439-0531.2012.02128.x.
[4] BR?NDLI SP. Long-term effect of repeated deslorelin acetate treatment in bitches for reproduction control.[J]. Theriogenology, 2021: 73-82. DOI:10.1016/j.theriogenology.2021.07.015.

Deslorelin acetate Preparation Products And Raw materials

Raw materials

Preparation Products

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View Lastest Price from Deslorelin acetate manufacturers

Nantong Guangyuan Chemicl Co,Ltd
Product
Deslorelin Acetate 82318-06-7
Price
US $10.00/kg
Min. Order
1kg
Purity
99%
Supply Ability
1000kg
Release date
2023-11-15

82318-06-7, Deslorelin acetateRelated Search:


  • 6-D-Tryptophan-9-(N-ethyl-L-prolinaMide)-1-9-luteinizing HorMone-releasing Factor (Swine) Monoacetate
  • BacheM 9022 Acetate
  • D-Trp LHRH-PEA Acetate
  • D-Trp6-Pro9-N-ethylaMide-LH-RH Acetate
  • H 4065 Acetate
  • PTL 3001 Acetate
  • SoMagard Aceta
  • Deslorelin Acetate(acetate)
  • 82318-06-7
  • C66H87N17O14
  • Amines
  • Aromatics
  • Chiral Reagents
  • Heterocycles
  • Intermediates & Fine Chemicals
  • Pharmaceuticals