6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-[1,2,4]triazolo[1,5-a]pyridine
- Product Name
- 6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-[1,2,4]triazolo[1,5-a]pyridine
- CAS No.
- 1160790-18-0
- Chemical Name
- 6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-[1,2,4]triazolo[1,5-a]pyridine
- Synonyms
- [1,2,4]Triazolo[1,5-a]pyridine-6-boronic acid pinacol ester;[1,2,4]TRIAZOLO[1,5-A]PYRIDIN-6-YLBORONIC ACID PINACOL ESTER;[1,2,4]Triazolo[1,5-a]pyridine-6-boronic acid pinacol ester 95%;[1,2,4]Triazolo[1,5-a]pyridine-6-boronic acid pinacol ester;6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-[1,2,4]triazolo[1,5-a]pyridine;[1,2,4]Triazolo[1,5-a]pyridine, 6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-
- CBNumber
- CB22520227
- Molecular Formula
- C12H16BN3O2
- Formula Weight
- 245.09
- MOL File
- 1160790-18-0.mol
6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-[1,2,4]triazolo[1,5-a]pyridine Property
- Melting point:
- 109-114°C
- Density
- 1.19±0.1 g/cm3(Predicted)
- storage temp.
- 2-8°C
- pka
- 2.71±0.30(Predicted)
- form
- solid
- Appearance
- White to off-white Solid
- InChI
- 1S/C12H16BN3O2/c1-11(2)12(3,4)18-13(17-11)9-5-6-10-14-8-15-16(10)7-9/h5-8H,1-4H3
- InChIKey
- QXPSJGKDBGYOEX-UHFFFAOYSA-N
- SMILES
- CC1(C)OB(OC1(C)C)c2ccc3ncnn3c2
Safety
- WGK Germany
- 3
- Storage Class
- 13 - Non Combustible Solids
N-Bromosuccinimide Price
- Product number
- T302823
- Product name
- 6-(4,4,5,5-Tetramethyl-1,3,2-dioxaborolan-2-yl)-[1,2,4]triazolo[1,5-a]pyridine
- Packaging
- 100mg
- Price
- $60
- Updated
- 2021/12/16
- Product number
- X5667
- Product name
- 6-(4,4,5,5-Tetramethyl-1,3,2-dioxaborolan-2-yl)[1,2,4]triazolo[1,5-a]pyridine
- Packaging
- 100mg
- Price
- $166
- Updated
- 2021/12/16
- Product number
- BOR0007060
- Product name
- 6-(4,4,5,5-TETRAMETHYL-1,3,2-DIOXABOROLAN-2-YL)-[1,2,4]-TRIAZOLO-[1,5-A]PYRIDINE
- Purity
- 95.00%
- Packaging
- 5MG
- Price
- $504.41
- Updated
- 2021/12/16
- Product number
- 143909
- Product name
- 6-(4,4,5,5-Tetramethyl-1,3,2-dioxaborolan-2-yl)-[1,2,4]triazolo[1,5-a]pyridine
- Purity
- 95%
- Packaging
- 1g
- Price
- $637
- Updated
- 2021/12/16
- Product number
- BOR0007060
- Product name
- 6-(4,4,5,5-TETRAMETHYL-1,3,2-DIOXABOROLAN-2-YL)-[1,2,4]-TRIAZOLO-[1,5-A]PYRIDINE
- Purity
- 95.00%
- Packaging
- 1G
- Price
- $825.3
- Updated
- 2021/12/16
6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-[1,2,4]triazolo[1,5-a]pyridine Chemical Properties,Usage,Production
Synthesis
356560-80-0
73183-34-3
1160790-18-0
6-Bromo-[1,2,4]triazolo[1,5-A]pyridine (180 mg, 0.91 mmol) and pinacol ester of biphenylboronic acid (348 mg, 1.37 mmol) were added 1,1'-bis(diphenylphosphino)ferrocene palladium(II) (37 mg, 0.045 mmol) and potassium acetate (180 mg, 1.83 mmol) in tetrahydrofuran (10 mL). The reaction was carried out at 80 °C for 8 h under nitrogen protection. After completion of the reaction, it was cooled to room temperature, filtered through diatomaceous earth and the solvent was evaporated under reduced pressure to afford [1,2,4]triazolo[1,5-a]pyridine-6-boronic acid pinacol ester (300 mg, yield: 74%).
References
[1] Patent: CN105254613, 2016, A. Location in patent: Paragraph 0349; 0350; 0351
[2] Patent: WO2009/74812, 2009, A1. Location in patent: Page/Page column 36
[3] Patent: WO2010/20363, 2010, A1. Location in patent: Page/Page column 87-88
6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-[1,2,4]triazolo[1,5-a]pyridine Preparation Products And Raw materials
Raw materials
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View Lastest Price from 6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-[1,2,4]triazolo[1,5-a]pyridine manufacturers
- Product
- 6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-[1,2,4]triazolo[1,5-a]pyridine 1160790-18-0
- Price
- US $1.00/KG
- Min. Order
- 1KG
- Purity
- 99%
- Supply Ability
- 100KG
- Release date
- 2019-12-23