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Cariprazine D8

Product Name
Cariprazine D8
CAS No.
1308278-50-3
Chemical Name
Cariprazine D8
Synonyms
Cariprazine D8;[2H8]-Cariprazine;Cariprazine D8 (Piperazine-d8);Cariprazine-D8 solution
CBNumber
CB23129380
Molecular Formula
C21H32Cl2N4O
Formula Weight
427.41
MOL File
1308278-50-3.mol
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Cariprazine D8 Property

Melting point:
>198°C (dec.)
storage temp. 
-20°C Freezer, Under inert atmosphere
solubility 
DMSO (Slightly), Methanol (Slightly)
form 
Solid
color 
Off-White to Pale Beige
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Hazard and Precautionary Statements (GHS)

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N-Bromosuccinimide Price

A2B
Product number
AX33668
Product name
Cariprazine-d8
Packaging
2.5mg
Price
$326
Updated
2021/12/16
A2B
Product number
AX33668
Product name
Cariprazine-d8
Packaging
10mg
Price
$776
Updated
2021/12/16
A2B
Product number
AX33668
Product name
Cariprazine-d8
Packaging
25mg
Price
$1536
Updated
2021/12/16
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Cariprazine D8 Chemical Properties,Usage,Production

Uses

Cariprazine-d8 is a deuterium labeled Cariprazine. Cariprazine is a novel antipsychotic agent candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate affinity for the 5-HT1A receptor (Ki=2.6 nM).

IC 50

D3 Receptor

References

[1] Seneca N, et al. Occupancy of dopamine D2 and D3 and serotonin 5-HT1A receptors by the novel antipsychotic drug candidate, cariprazine (RGH-188), in monkey brain measured using positron emission tomography. Psychopharmacology (Berl). 2011 Dec;218(3):579-8. DOI:10.1007/s00213-011-2343-z

Cariprazine D8 Preparation Products And Raw materials

Raw materials

Preparation Products

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Cariprazine D8 Suppliers

China 7 India 4 United States 1 Global 12
Shanghai Champ Biopharmaceuticals Co., Ltd.
Tel
021-61537865 13585780846
Email
sales@champchem.com
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China
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Zhengzhou Acme Chemical Co., Ltd.
Tel
0371-037163312495,13303845143 13303845143
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QQ3001379618
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3001379618@qq.com
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China
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10267
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BOC Sciences
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+1-631-485-4226
Fax
1-631-614-7828
Email
inquiry@bocsci.com
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United States
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19552
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Manhag Testing Technology Co., Ltd
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020-3846 2365 19110442770
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458677837@qq.com
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China
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7775
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Nanjing Shizhou Biology Technology Co.,Ltd
Tel
17301488900
Fax
025-85560043
Email
judy.xia@synzest.com
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China
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12582
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BePure (Beijing) Biotechnology Co.
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58896805
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7993601name@qq.com
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CHINA
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6620
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Merck KGaA
Tel
21-20338288
Email
ordercn@merckgroup.com
Country
China
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1308278-50-3, Cariprazine D8Related Search:

Cariprazine Nsc175383 Cariprazine intermediate 2 Desmethyl Cariprazine Piperazine, 1-(2-chloroethyl)-4-(2,3-dichlorophenyl)- Urea, N,N'-bis[trans-4-[2-[4-(2,3-dichlorophenyl)-1-piperazinyl]ethyl]cyclohexyl]- Urea, N,N-dimethyl-N'-[trans-4-[2-[[(4-methylphenyl)sulfonyl]oxy]ethyl]cyclohexyl]- ethyl dimethylcarbamate 3,3-dimethyl-1-[(1r,4r)-4-(2-hydroxyethyl)cyclohexyl]urea Cyclohexaneethanol, 4-amino-, hydrochloride (1:1), trans-

  • Cariprazine D8
  • [2H8]-Cariprazine
  • Cariprazine D8 (Piperazine-d8)
  • Cariprazine-D<sub>8</sub> solution
  • 1308278-50-3