BI-3802

Product Name: BI-3802
CAS No.: 2166387-65-9
Chemical Name: BI-3802
Synonyms: BI-3802;BI-3802 ，S6937;BI-3802 (BI3802;BI-3802, 10 mM in DMSO;Inhibitor,Bcl-2 Family,BI3802,BI-3802,BI 3802,inhibit;cis-2-((6-((5-chloro-2-(3,5-dimethylpiperidin-1-yl)pyrimidin-4-yl)amino)-1-methyl-2-oxo-1,2-dihydroquinolin-3-yl)oxy)-N-methylacetamide;Acetamide, 2-[[6-[[5-chloro-2-[(3R,5S)-3,5-dimethyl-1-piperidinyl]-4-pyrimidinyl]amino]-1,2-dihydro-1-methyl-2-oxo-3-quinolinyl]oxy]-N-methyl-, rel-
CBNumber: CB24667636
Molecular Formula: C24H29ClN6O3
Formula Weight: 484.98
MOL File: 2166387-65-9.mol

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BI-3802 Property

Density: 1.35±0.1 g/cm3(Predicted)
storage temp.: Store at -20°C
solubility: DMSO : 5 mg/mL (10.31 mM);Methanol : 2 mg/mL (4.12 mM; ultrasonic and adjust pH to 5 with 1M HCl);Water : < 0.1 mg/mL (insoluble)
form: Solid
pka: 14.74±0.46(Predicted)
color: White to off-white

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Hazard and Precautionary Statements (GHS)

Symbol(GHS)

Signal word

Warning

Hazard statements

H302Harmful if swallowed

H315Causes skin irritation

H319Causes serious eye irritation

H335May cause respiratory irritation

Precautionary statements

P261Avoid breathing dust/fume/gas/mist/vapours/spray.

P305+P351+P338IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses, if present and easy to do. Continuerinsing.

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N-Bromosuccinimide Price

Sigma-Aldrich

Product number: SML4079
Product name: BI-3802
Purity: ≥98% (HPLC)
Packaging: 1 unit
Price: $479
Updated: 2025/07/31

Axon Medchem

Product number: Axon3361
Product name: BI-3802
Purity: 99%
Packaging: 25mg
Price: $979
Updated: 2021/12/16

Axon Medchem

Product number: Axon3361
Product name: BI-3802
Purity: 99%
Packaging: 2mg
Price: $143
Updated: 2021/12/16

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BI-3802 Chemical Properties,Usage,Production

Uses

BI-3802 is a highly potent BCL6 degrader and inhibits the Bric-à-brac (BTB) domain of BCL6 with an IC50 of ≤3 nM. BI-3802 induces the polymerization of BCL6 and promotes BCL6 degration depended on E3 ligase SIAH1. BI-3802 has antitumor activity[1][2].

References

[1] Kerres N, et al. Chemically Induced Degradation of the Oncogenic Transcription Factor BCL6. Cell Rep. 2017 Sep 19;20(12):2860-2875. DOI:10.1016/j.celrep.2017.08.081
[2] Miko?aj S?abicki, et al. Small-molecule-induced polymerization triggers degradation of BCL6. Nature. 2020 Nov 18. DOI:10.1038/s41586-020-2925-1

BI-3802 Preparation Products And Raw materials

Raw materials

Preparation Products

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BI-3802 Suppliers

China 46 United States 4 Global 50

Beijing HwrkChemical Technology Co., Ltd

Tel: 18515581800 18501085097
Fax: 010-89508210
Email: sales.bj@hwrkchemical.com
Country: China
ProdList: 9400
Advantage: 55

BOC Sciences

Tel: 1-631-485-4226; 16314854226
Email: info@bocsci.com
Country: United States
ProdList: 12952
Advantage: 65

Shanghai Raise Chemical Technology Co.,Ltd

Tel: 15026594951
Fax: 0556-5030632
Email: rs@raise-chem.com
Country: China
ProdList: 4454
Advantage: 55

ShangHai Caerulum Pharma Discovery Co., Ltd.

Tel: 18149758185
Email: sales-cpd@caerulumpharma.com
Country: China
ProdList: 3506
Advantage: 58

Shanghai EFE Biological Technology Co., Ltd.

Tel: 021-65675885 18964387627
Fax: 021-65675885
Email: info@efebio.com
Country: China
ProdList: 9803
Advantage: 58

Shanghai YuanYe Biotechnology Co., Ltd.

Tel: 021-61312847; 18021002903
Fax: QQ:3008007432
Email: 3008007409@qq.com
Country: China
ProdList: 71826
Advantage: 60

Wellman Pharmaceutical Group Limited

Tel: 027-027-83778875 15807197853
Fax: 027-83991220
Email: 15807197853@163.com
Country: China
ProdList: 3932
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Shanghai Akasaka Biotechnology Co., Ltd.

Tel: 15121162054
Country: CHINA
ProdList: 635
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Jilin Province Woda Biotechnology Co., Ltd.

Tel: 13504435624
Email: 1927928688@qq.com
Country: China
ProdList: 1615
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TargetMol Chemicals Inc.

Tel: +1-781-999-5354; +17819995354
Email: marketing@targetmol.com
Country: United States
ProdList: 32435
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2166387-65-9, BI-3802Related Search:

BI-3802

BI-3802 (BI3802

cis-2-((6-((5-chloro-2-(3,5-dimethylpiperidin-1-yl)pyrimidin-4-yl)amino)-1-methyl-2-oxo-1,2-dihydroquinolin-3-yl)oxy)-N-methylacetamide

Inhibitor,Bcl-2 Family,BI3802,BI-3802,BI 3802,inhibit

Acetamide, 2-[[6-[[5-chloro-2-[(3R,5S)-3,5-dimethyl-1-piperidinyl]-4-pyrimidinyl]amino]-1,2-dihydro-1-methyl-2-oxo-3-quinolinyl]oxy]-N-methyl-, rel-

BI-3802, 10 mM in DMSO

BI-3802 ，S6937

2166387-65-9