ChemicalBook > CAS DataBase List > 5-(BROMOMETHYL)-2-METHOXYPYRIDINE

5-(BROMOMETHYL)-2-METHOXYPYRIDINE

Product Name
5-(BROMOMETHYL)-2-METHOXYPYRIDINE
CAS No.
128632-03-1
Chemical Name
5-(BROMOMETHYL)-2-METHOXYPYRIDINE
Synonyms
5-(BROMOMETHYL)-2-METHOXYPYRIDINE;Pyridine, 5-(bromomethyl)-2-methoxy-
CBNumber
CB32459717
Molecular Formula
C7H8BrNO
Formula Weight
202.05
MOL File
128632-03-1.mol
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5-(BROMOMETHYL)-2-METHOXYPYRIDINE Property

Boiling point:
249.0±25.0 °C(Predicted)
Density 
1.484±0.06 g/cm3(Predicted)
storage temp. 
under inert gas (nitrogen or Argon) at 2-8°C
pka
2.49±0.10(Predicted)
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Hazard and Precautionary Statements (GHS)

Symbol(GHS)
Signal word
Warning
Hazard statements

H303May be harmfulif swallowed

H320Causes eye irritation

Precautionary statements

P264Wash hands thoroughly after handling.

P264Wash skin thouroughly after handling.

P305+P351+P338IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses, if present and easy to do. Continuerinsing.

P312Call a POISON CENTER or doctor/physician if you feel unwell.

P337+P313IF eye irritation persists: Get medical advice/attention.

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N-Bromosuccinimide Price

AK Scientific
Product number
Y7368
Product name
5-(Bromomethyl)-2-methoxypyridine
Packaging
250mg
Price
$192
Updated
2021/12/16
Chemenu
Product number
CM248697
Product name
5-(Bromomethyl)-2-methoxypyridine
Purity
95%
Packaging
1g
Price
$248
Updated
2021/12/16
Ambeed
Product number
A180366
Product name
5-(Bromomethyl)-2-methoxypyridine
Purity
95%
Packaging
1g
Price
$287
Updated
2021/12/16
Crysdot
Product number
CD11300264
Product name
5-(Bromomethyl)-2-methoxypyridine
Purity
95+%
Packaging
1g
Price
$325
Updated
2021/12/16
Chemenu
Product number
CM248697
Product name
5-(Bromomethyl)-2-methoxypyridine
Purity
95%
Packaging
5g
Price
$842
Updated
2021/12/16
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5-(BROMOMETHYL)-2-METHOXYPYRIDINE Chemical Properties,Usage,Production

Synthesis

58584-63-7

128632-03-1

(6-Methoxypyridin-3-yl)methanol (250 mg, 1.797 mmol, commercially available from e.g. Fluorochem) was used as starting material, which was dissolved in chloroform (20 mL) in a 50 mL round bottom flask. Phosphorus tribromide (0.188 mL, 1.989 mmol) was slowly added dropwise to the reaction system at 0 °C. After the reaction was completed, the reaction was stopped and the reaction was completed. After the dropwise addition, the reaction mixture was stirred at room temperature for 1 hour. After completion of the reaction, the reaction mixture was washed with water (3 x 30 mL) and the organic layer was separated. The organic phases were combined, washed with saturated saline (30 mL), filtered through a hydrophobic glass stock and concentrated under reduced pressure to remove the solvent. The resulting oily crude product was dissolved in dichloromethane and purified by column chromatography on a Biage Isolera SNAP 25g silica gel with an elution gradient of 0-4% cyclohexane/ethyl acetate. The fraction containing the target product was collected and concentrated under reduced pressure to give 5-(bromomethyl)-2-methoxypyridine (160 mg, 0.792 mmol, 44% yield) as a colorless oil.The results of LCMS (2 mM formic acid) analysis were: retention time (Rt) = 0.93 min, [M+H]+ = 202.

References

[1] Journal of Labelled Compounds and Radiopharmaceuticals, 2007, vol. 50, # 5-6, p. 613 - 615
[2] Patent: WO2017/37116, 2017, A1. Location in patent: Page/Page column 76

5-(BROMOMETHYL)-2-METHOXYPYRIDINE Preparation Products And Raw materials

Raw materials

Preparation Products

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5-(BROMOMETHYL)-2-METHOXYPYRIDINE Suppliers

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128632-03-1, 5-(BROMOMETHYL)-2-METHOXYPYRIDINERelated Search:


  • 5-(BROMOMETHYL)-2-METHOXYPYRIDINE
  • Pyridine, 5-(bromomethyl)-2-methoxy-
  • 128632-03-1