ChemicalBook > CAS DataBase List > (±)17-HETE

(±)17-HETE

Product Name
(±)17-HETE
CAS No.
128914-47-6
Chemical Name
(±)17-HETE
Synonyms
(±)17-HETE;OPPIPPRXLIDJKN-JPURVOHMSA-N;17-hydroxy-5(Z),8(Z),11(Z),14(Z)-ETA;17-hydroxy-5(Z),8(Z),11(Z),14(Z)-eicosatetraenoic acid;5,8,11,14-Eicosatetraenoic acid, 17-hydroxy-, (5Z,8Z,11Z,14Z)-
CBNumber
CB32589795
Molecular Formula
C20H32O3
Formula Weight
320.47
MOL File
128914-47-6.mol
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(±)17-HETE Property

storage temp. 
Store at -20°C
solubility 
0.1 m Na2CO3: 2 mg/ml; DMF: Miscible; DMSO: Miscible; Ethanol: Miscible; PBS (pH 7.2): 0.8 mg/ml
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Hazard and Precautionary Statements (GHS)

Symbol(GHS)
Signal word
Danger
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N-Bromosuccinimide Price

Cayman Chemical
Product number
10010636
Product name
(±)17-HETE
Purity
≥98%
Packaging
25μg
Price
$146
Updated
2024/03/01
Cayman Chemical
Product number
10010636
Product name
(±)17-HETE
Purity
≥98%
Packaging
50μg
Price
$278
Updated
2024/03/01
Cayman Chemical
Product number
10010636
Product name
(±)17-HETE
Purity
≥98%
Packaging
100μg
Price
$525
Updated
2024/03/01
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(±)17-HETE Chemical Properties,Usage,Production

Description

Electrolyte and fluid transport in the kidney are regulated in part by arachidonic acid and its metabolites. (±)17-HETE is the racemic version of a cytochrome P450 (CYP450) metabolite of arachidonic acid that has stereospecific effects on sodium transport in the kidney. At a concentration of 2 μM the (S)-enantiomer of 17-HETE inhibits proximal tubule ATPase activity by as much as 70%, whereas the (R)-isomer is inactive.

Uses

17-HETE is arachidonic acid metabolite through cytochrome P-450 pathways, which consists of 17R-HETE and 17S-HETE enantiomers. 17-HETE serves as allosteric activator of the cytochrome P450 1B1 and inhibitor of ATPase, induces cardic hypertrophy[1][2].

Definition

ChEBI: A HETE that consists of arachidonic acid bearing an additional hydroxy substituent at position 17.

in vivo

17-HETE (1-20 μg, i.a.) stereospecificially inhibits proximal tubule ATPase activity with S- enantiomer in New Zealand white rabbit[2].

Animal Model:New Zealand White rabbit[2]
Dosage:1-20 μg
Administration:injection into artery
Result:17S inhibited more than 70% ATPase activity at the concentration of 2 μM, while 17R enantiomer remained inactive.

IC 50

CYP1B1

References

[1] Isse FA, et al., 17-(R/S)-hydroxyeicosatetraenoic acid (HETE) induces cardiac hypertrophy through the CYP1B1 in enantioselective manners. Prostaglandins Other Lipid Mediat. 2023 Oct;168:106749. DOI:10.1016/j.prostaglandins.2023.106749
[2] Carroll MA, e al., Cytochrome P-450-dependent HETEs: profile of biological activity and stimulation by vasoactive peptides. Am J Physiol. 1996 Oct;271(4 Pt 2):R863-9. DOI:10.1152/ajpregu.1996.271.4.R863

(±)17-HETE Preparation Products And Raw materials

Raw materials

Preparation Products

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(±)17-HETE Suppliers

BOC Sciences
Tel
1-631-485-4226; 16314854226
Email
info@bocsci.com
Country
United States
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12952
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Yichang Zhongyitai Trading Co., Ltd.
Tel
0717-6449896 13886658719
Fax
0717-6558598
Email
root@zhongyitai.com
Country
China
ProdList
1978
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Alfa Chemistry
Tel
1-516-6625404
Fax
1-516-927-0118
Email
support@alfa-chemistry.com
Country
United States
ProdList
9171
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Shanghai Hongye Biotechnology Co. Ltd
Tel
400-9205774
Email
sales@glpbio.cn
Country
China
ProdList
6777
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58
ChemeGen(Shanghai) Biotechnology Co.,Ltd.
Tel
18818260767
Fax
QQ 3610331285
Email
sales@chemegen.com
Country
China
ProdList
11218
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58
MedBioPharmaceutical Technology Inc
Tel
021-69568360 18916172912
Email
order@med-bio.cn
Country
China
ProdList
8140
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58
amyjet
Tel
4006800868;027-59626688 18371453821;18771149750
Email
sales@amyjet.com
Country
China
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2917
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58
TargetMol Chemicals Inc.
Tel
4008200310
Email
marketing@tsbiochem.com
Country
China
ProdList
24964
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Shanghai Yifei Biotechnology Co. , Ltd.
Tel
021-65675885 18964387627
Email
customer_service@efebio.com
Country
China
ProdList
11973
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58
SHANGHAI ZZBIO CO., LTD.
Tel
15102117276 19921389125
Email
tech@zzbioco.com
Country
China
ProdList
12064
Advantage
58

128914-47-6, (±)17-HETERelated Search:


  • (±)17-HETE
  • OPPIPPRXLIDJKN-JPURVOHMSA-N
  • 5,8,11,14-Eicosatetraenoic acid, 17-hydroxy-, (5Z,8Z,11Z,14Z)-
  • 17-hydroxy-5(Z),8(Z),11(Z),14(Z)-eicosatetraenoic acid
  • 17-hydroxy-5(Z),8(Z),11(Z),14(Z)-ETA
  • 128914-47-6