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CAY10498

Product Name
CAY10498
CAS No.
863202-33-9
Chemical Name
CAY10498
Synonyms
CAY10498;A3AR antagonist 3;CAY10498,CAY-10498;2-phenyl-amino-N6-endo-norbornyladenine;CAY10498, A3 adenosine receptor antagonist;6-N-(3-bicyclo[2.2.1]heptanyl)-2-N-phenyl-7H-purine-2,6-diamine;1H-Purine-2,6-diamine, N6-(1R,2S,4S)-bicyclo(2.2.1)hept-2-yl-N2-phenyl;9H-Purine-2,6-diamine, N6-(1R,2S,4S)-bicyclo[2.2.1]hept-2-yl-N2-phenyl-, rel-
CBNumber
CB32590412
Molecular Formula
C18H20N6
Formula Weight
320.39
MOL File
863202-33-9.mol
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CAY10498 Property

Boiling point:
652.0±58.0 °C(Predicted)
Density 
1.403±0.06 g/cm3(Predicted)
storage temp. 
Store at -20°C
solubility 
DMF: 10 mg/ml; DMSO: 10 mg/ml; DMSO:PBS (pH 7.2) (1:4): .2 mg/ml; Ethanol: 1 mg/ml
form 
A crystalline solid
pka
10.63±0.10(Predicted)
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Hazard and Precautionary Statements (GHS)

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N-Bromosuccinimide Price

Cayman Chemical
Product number
10007955
Product name
CAY10498
Purity
≥95%
Packaging
500μg
Price
$121
Updated
2024/03/01
Cayman Chemical
Product number
10007955
Product name
CAY10498
Purity
≥95%
Packaging
1mg
Price
$218
Updated
2024/03/01
Cayman Chemical
Product number
10007955
Product name
CAY10498
Purity
≥95%
Packaging
5mg
Price
$961
Updated
2024/03/01
American Custom Chemicals Corporation
Product number
NUC0002272
Product name
1H-PURINE-2,6-DIAMINE, N6-(1R,2S,4S)-BICYCLO(2.2.1)HEPT-2-YL-N2-PHENYL
Purity
95.00%
Packaging
5MG
Price
$502.99
Updated
2021/12/16
AK Scientific
Product number
1287AH
Product name
1H-Purine-2,6-diamine,N6-(1R,2S,4S)-bicyclo(2.2.1)hept-2-yl-N2-phenyl
Packaging
5mg
Price
$1169
Updated
2021/12/16
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CAY10498 Chemical Properties,Usage,Production

Uses

A3AR antagonist 3 (compound 21) is a selective A3 adenosine receptor (A3AR) antagonist with a Ki of 37 nM. A3AR antagonist 3 shows >60-fold selectivity in comparison to A1 and A2A adenosine receptors[1].

IC 50

hA3: 37 nM (Ki); hA1AR: 2.22 μM (Ki); hA2AAR: 7.73 μM (Ki)

References

[1] Melissa Perreira, et al. "Reversine" and its 2-substituted adenine derivatives as potent and selective A3 adenosine receptor antagonists. J Med Chem. 2005 Jul 28;48(15):4910-8. DOI:10.1021/jm050221l

CAY10498 Preparation Products And Raw materials

Raw materials

Preparation Products

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CAY10498 Suppliers

China 32 United States 6 Global 38
BOC Sciences
Tel
1-631-485-4226; 16314854226
Email
info@bocsci.com
Country
United States
ProdList
12952
Advantage
65
BOC Sciences
Tel
16314854226
Email
info@bocsci.com
Country
United States
ProdList
9923
Advantage
65
Shanghai EFE Biological Technology Co., Ltd.
Tel
021-65675885 18964387627
Fax
021-65675885
Email
info@efebio.com
Country
China
ProdList
9803
Advantage
58
Shanghai Hongye Biotechnology Co. Ltd
Tel
400-9205774
Email
sales@glpbio.cn
Country
China
ProdList
6777
Advantage
58
TargetMol Chemicals Inc.
Tel
+1-781-999-5354; +17819995354
Email
marketing@targetmol.com
Country
United States
ProdList
32470
Advantage
58
ChemeGen(Shanghai) Biotechnology Co.,Ltd.
Tel
18818260767
Fax
QQ 3610331285
Email
sales@chemegen.com
Country
China
ProdList
11218
Advantage
58
Taizhou Nanfeng Pharmaceutical Research Institute
Tel
nanfengdrug@163.com; 18616377689
Email
nanfengdrug@163.com
Country
China
ProdList
20009
Advantage
58
TargetMol Chemicals Inc.
Tel
4008200310
Email
marketing@tsbiochem.com
Country
China
ProdList
24964
Advantage
58
Cayman Chemical Company
Tel
800-364-9897
Email
sales@caymanchem.com
Country
China
ProdList
6838
Advantage
58
Biosynth Biological Technology (Suzhou) Co Ltd
Tel
51288865780
Email
sales@biosynth.com
Country
China
ProdList
6051
Advantage
58

863202-33-9, CAY10498Related Search:


  • CAY10498
  • 2-phenyl-amino-N6-endo-norbornyladenine
  • 6-N-(3-bicyclo[2.2.1]heptanyl)-2-N-phenyl-7H-purine-2,6-diamine
  • 9H-Purine-2,6-diamine, N6-(1R,2S,4S)-bicyclo[2.2.1]hept-2-yl-N2-phenyl-, rel-
  • CAY10498,CAY-10498
  • A3AR antagonist 3
  • CAY10498, A3 adenosine receptor antagonist
  • 1H-Purine-2,6-diamine, N6-(1R,2S,4S)-bicyclo(2.2.1)hept-2-yl-N2-phenyl
  • 863202-33-9